SCHEMBL3928065

SCHEMBL3928065

Oc1ccc2nc(-c3cc(F)c(O)c(F)c3)c(Br)cc2c1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 15/20 0.59
ESR1 P03372 14/20 0.59
RPS6KA3 P51812 2/20 0.39
ESRRB O95718 1/20 0.38
ESRRA P11474 1/20 0.38
PDE3B Q13370 1/20 0.37
PDE3A Q14432 1/20 0.37
GPBAR1 Q8TDU6 1/20 0.36
DHODH Q02127 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3922895 0.82 ESR2 (0.51) ESR2ESR1ESRRBESRRAPDE3B
SCHEMBL3928207 0.75 ESR1 (1.00) ESR2ESR1ESRRBESRRA
SCHEMBL27905510 0.71 PDE3B (0.46) ESR2ESR1ESRRBESRRAPDE3B
SCHEMBL27638492 0.69 ESR2 (0.43) ESR2ESR1
SCHEMBL28211226 0.68 ESR1 (0.42) ESR2ESR1ESRRBESRRAPDE3B
SCHEMBL3934682 0.66 ESR1 (1.00) ESR2ESR1
SCHEMBL3044443 0.66 ESR2 (0.54) ESR2ESR1PDE3BPDE3A
SCHEMBL1289652 0.65 KDM4E (0.50) DHODH
SCHEMBL3557738 0.65 PIM1 (0.43) ESR2ESR1ESRRBESRRAPDE3B
SCHEMBL15552163 0.64 ESR1 (0.48) ESR2ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009417-A2 PHARMACEUTICAL COMPOSITIONS AND METHODS OF PREVENTING, TREATING, OR INHIBITING INFLAMMATORY DISEASES, DISORDERS, OR CONDITIONS OF THE SKIN, AND DISEASES, DISORDERS, OR CONDITIONS ASSOCIATED WITH COLLAGEN DEPLETION WYETH (US) 2009-01-15 WO disclosed