SCHEMBL3928091

SCHEMBL3928091

NC=CC(c1ccccc1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.43
F2 P00734 1/20 0.43
TAAR1 Q96RJ0 3/20 0.40
HTR2A P28223 1/20 0.40
TSHR P16473 1/20 0.38
HRH1 P35367 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
ADRA2A P08913 1/20 0.34
ADRA2C P18825 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3928088 1.00 DPP4 (0.43) DPP4F2TAAR1HTR2ATSHR
Hydrochloric Acid SCHEMBL7317204 0.97 DPP4 (0.42) DPP4F2TAAR1HTR2ATSHR
SCHEMBL8522965 0.83 DPP4 (0.45) DPP4F2TAAR1HTR2ATSHR
SCHEMBL9804521 0.80 ACP3 (0.42) HTR2AHRH1SLC6A2SLC6A4SLC6A3
SCHEMBL6014583 0.75 TRPA1 (0.44) DPP4F2TAAR1ADRA2AADRA2C
SCHEMBL6014580 0.75 TRPA1 (0.44) DPP4F2TAAR1ADRA2AADRA2C
SCHEMBL8613849 0.74 MEN1 (0.39) DPP4F2TAAR1HTR2ATSHR
SCHEMBL692130 0.74 MEN1 (0.39) DPP4F2TAAR1HTR2ATSHR
SCHEMBL2387572 0.74 DPP4 (0.38) DPP4F2TAAR1HTR2ATSHR
SCHEMBL2094186 0.74 CYP2D6 (0.39) DPP4F2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE40851-E1 3,3-diphenylpropylamines, their use and preparation PFIZER HEALTH AB (SE) 2009-07-14 US claimed
US-RE39667-E1 3,3-Diphenylpropylamines, their use and preparation PFIZER HEALTH AB (SE) 2007-05-29 US claimed
EP-0667852-B1 NOVEL 3,3-DIPHENYLPROPYLAMINES, THEIR USE AND PREPARATION PHARMACIA & UPJOHN AB (SE) 1998-04-08 EP claimed
US-5559269-A ANTICHOLINERGIC AGENTS PHARMACIA AB (SE) 1996-09-24 US claimed
EP-0667852-A1 NOVEL 3,3-DIPHENYLPROPYLAMINES, THEIR USE AND PREPARATION Pharmacia & Upjohn Aktiebolag (SE) 1995-08-23 EP claimed
WO-1994011337-A9 NOVEL 3,3-DIPHENYLPROPYLAMINES, THEIR USE AND PREPARATION 1995-07-06 WO claimed
WO-1994011337-A1 NOVEL 3,3-DIPHENYLPROPYLAMINES, THEIR USE AND PREPARATION PHARMACIA AB (SE) 1994-05-26 WO claimed
CN-105074514-A Polarizing plate SUMITOMO CHEMICAL CO 2015-11-18 CN disclosed
US-RE40851-E1 3,3-diphenylpropylamines, their use and preparation PFIZER HEALTH AB (SE) 2009-07-14 US disclosed
US-RE39667-E1 3,3-Diphenylpropylamines, their use and preparation PFIZER HEALTH AB (SE) 2007-05-29 US disclosed
EP-1534239-A2 PREPARATION OF SUBMICRON SIZED PARTICLES WITH POLYMORPH CONTROL AND NEW POLYMORPH OF ITRACONAZOLE BAXTER INTERNATIONAL INC. (US) 2005-06-01 EP disclosed
WO-2004054500-A2 PREPARATION OF SUBMICRON SIZED PARTICLES WITH POLYMORPH CONTROL AND NEW POLYMORPH OF ITRACONAZOLE BAXTER INTERNATIONAL INC. (US) 2004-07-01 WO disclosed
US-20030096013-A1 Preparation of submicron sized particles with polymorph control BAXTER INTERNATIONAL INC. 2003-05-22 US disclosed
EP-0667852-B1 NOVEL 3,3-DIPHENYLPROPYLAMINES, THEIR USE AND PREPARATION PHARMACIA & UPJOHN AB (SE) 1998-04-08 EP disclosed
US-5686464-A ANTICHOLINERGIC AGENTS; URINARY INCONTINENCE TREATMENT PHARMACIA AB (SE) 1997-11-11 US disclosed
US-5559269-A ANTICHOLINERGIC AGENTS PHARMACIA AB (SE) 1996-09-24 US disclosed
EP-0667852-A1 NOVEL 3,3-DIPHENYLPROPYLAMINES, THEIR USE AND PREPARATION Pharmacia & Upjohn Aktiebolag (SE) 1995-08-23 EP disclosed
WO-1994011337-A9 NOVEL 3,3-DIPHENYLPROPYLAMINES, THEIR USE AND PREPARATION 1995-07-06 WO disclosed
WO-1994011337-A1 NOVEL 3,3-DIPHENYLPROPYLAMINES, THEIR USE AND PREPARATION PHARMACIA AB (SE) 1994-05-26 WO disclosed