SCHEMBL3928181

SCHEMBL3928181

CCCCOC(=O)N1CCN(c2nc3cc(C)ccc3o2)C(COc2cccnc2)C1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
KCNH2 Q12809 1/20 0.42
DRD2 P14416 3/20 0.39
DRD3 P35462 3/20 0.39
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3940090 0.88 CHRNA7 (0.47) CHRNA7CHRNB2CHRNA4KCNH2DRD2
SCHEMBL780477 0.87 GPR119 (0.44) CHRNA7CHRNB2CHRNA4KCNH2DRD2
SCHEMBL779655 0.81 GPR119 (0.44) CHRNA7CHRNB2CHRNA4KCNH2DRD2
SCHEMBL780438 0.78 CHRNA7 (0.47) CHRNA7CHRNB2CHRNA4KCNH2DRD2
SCHEMBL781787 0.77 CHRNA7 (0.44) CHRNA7CHRNB2CHRNA4KCNH2
SCHEMBL780001 0.76 CHRNA7 (0.71) CHRNA7CHRNB2CHRNA4KCNH2
SCHEMBL780000 0.76 CHRNA7 (0.71) CHRNA7CHRNB2CHRNA4KCNH2
Hydrochloric Acid SCHEMBL778801 0.75 CHRNA7 (0.71) CHRNA7CHRNB2CHRNA4KCNH2
Hydrochloric Acid SCHEMBL15841836 0.75 CHRNA7 (0.71) CHRNA7CHRNB2CHRNA4KCNH2
SCHEMBL780135 0.73 CHRNA7 (0.60) CHRNA7CHRNB2CHRNA4KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044038-A2 NOVEL PIPERAZINES, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE THEREOF Cornerstone Therapeutics Inc. (US) 2009-04-08 EP disclosed
WO-2007146066-A2 NOVEL PIPERAZINES, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE THEREOF CRITICAL THERAPEUTICS, INC. (US) 2007-12-21 WO disclosed