SCHEMBL3929189

SCHEMBL3929189

Cc1csc(S(=O)(=O)C2(c3cc(N4CCOCC4)nc(-c4ccc(NC(=O)Nc5c[nH]nc5C)cc4)n3)CC2)n1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ATR Q13535 7/20 0.44
PIK3CA P42336 13/20 0.44
MTOR P42345 11/20 0.44
PIK3CD O00329 3/20 0.43
PIK3CG P48736 9/20 0.41
PIK3CB P42338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3928892 0.88 MTOR (0.51) ATRPIK3CAMTORPIK3CDPIK3CG
SCHEMBL3936892 0.88 ATR (0.59) ATRPIK3CAMTORPIK3CD
SCHEMBL3927820 0.87 ATR (0.46) ATRPIK3CAMTORPIK3CDPIK3CG
SCHEMBL4197826 0.86 PIK3CA (0.59) ATRPIK3CAMTORPIK3CDPIK3CG
SCHEMBL3932956 0.86 ATR (0.48) ATRPIK3CAMTORPIK3CDPIK3CG
SCHEMBL3929187 0.85 ATR (0.46) ATRPIK3CAMTORPIK3CDPIK3CG
SCHEMBL3928847 0.85 ATR (0.47) ATRPIK3CAMTORPIK3CDPIK3CG
SCHEMBL3928570 0.84 PIK3CA (0.52) ATRPIK3CAMTORPIK3CDPIK3CG
SCHEMBL4203443 0.84 MTOR (0.51) ATRPIK3CAMTORPIK3CDPIK3CG
SCHEMBL3932917 0.84 ATR (0.46) ATRPIK3CAMTORPIK3CDPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074118-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES AstraZeneca AB (SE) 2009-07-01 EP disclosed
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed