SCHEMBL3930028

SCHEMBL3930028

CC(C)(C)N1CCN(C(=O)c2ccc(-c3ccccc3Cl)s2)C(COc2cccnc2)C1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHRNA1 P02708 1/20 0.38
CHRNB1 P11230 1/20 0.38
CHRNB2 P17787 1/20 0.38
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
CHRNB3 Q05901 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL778984 0.88 POLB (0.40) CHRNA1CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL778262 0.85 CHRNA7 (0.52) CHRNA7
Hydrochloric Acid SCHEMBL780024 0.84
SCHEMBL3928367 0.79 CHRNA7 (0.42) CHRNA1CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL3939831 0.78 CHRNA7 (0.41) CHRNA1CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL3939406 0.74 CHRNA7 (0.40) CHRNA1CHRNB1CHRNB2CHRNB4CHRNA3
SCHEMBL3932862 0.72 CHRNA7 (0.55) CHRNA7
SCHEMBL779154 0.72 CHRNA7 (0.51) CHRNA7
Hydrochloric Acid SCHEMBL778260 0.72 KCNH2 (0.56)
SCHEMBL780993 0.72 RECQL (0.43) CHRNA1CHRNB1CHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044038-A2 NOVEL PIPERAZINES, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE THEREOF Cornerstone Therapeutics Inc. (US) 2009-04-08 EP disclosed
WO-2007146066-A2 NOVEL PIPERAZINES, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE THEREOF CRITICAL THERAPEUTICS, INC. (US) 2007-12-21 WO disclosed