SCHEMBL3930877

SCHEMBL3930877

O=C(Cc1c(Cl)c(F)nc(F)c1Cl)OCc1ccccc1.O=C(O)Cc1c(Cl)c(F)nc(F)c1Cl

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
MAPK1 P28482 2/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
CASP1 P29466 2/20 0.43
PAM P19021 1/20 0.41
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39
PLAU P00749 3/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A3 Q01959 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ENPP2 Q13822 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL501799 0.96 ALDH1A1 (0.57) ALDH1A1MAPK1L3MBTL1CASP1PAM
SCHEMBL501448 0.90 ALDH1A1 (0.53) ALDH1A1MAPK1L3MBTL1CASP1PAM
SCHEMBL501844 0.78 AKR1B1 (0.42) ALDH1A1
SCHEMBL11852691 0.74 ALDH1A1 (0.66) ALDH1A1MAPK1L3MBTL1CASP1KMT2A
SCHEMBL502353 0.74 ELANE (0.52) ALDH1A1MAPK1L3MBTL1KMT2APOLB
SCHEMBL24464462 0.73 ALDH1A1 (0.41) ALDH1A1MAPK1L3MBTL1KMT2APOLB
SCHEMBL31245908 0.72 ALDH1A1 (0.85) ALDH1A1MAPK1L3MBTL1CASP1PAM
SCHEMBL16366728 0.72 ALDH1A1 (0.62) ALDH1A1MAPK1L3MBTL1PAMKMT2A
SCHEMBL10204657 0.71 ELANE (0.49) ALDH1A1MAPK1L3MBTL1KMT2APOLB
SCHEMBL361779 0.71 ALDH1A1 (1.00) ALDH1A1MAPK1L3MBTL1CASP1PAM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044037-A2 HIV REVERSE TRANSCRIPTASE INHIBITORS Gilead Sciences, Inc. (US) 2009-04-08 EP disclosed
WO-2008016522-A2 HIV REVERSE TRANSCRIPTASE INHIBITORS GILEAD SCIENCES, INC. (US) 2008-02-07 WO disclosed