SCHEMBL3931027

SCHEMBL3931027

COC(=O)Nc1cc(C(=O)c2ccnc(OC)c2)cc(-c2cccc3occc23)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.42
KCNK9 Q9NPC2 1/20 0.42
CNR1 P21554 1/20 0.38
PLCG1 P19174 1/20 0.35
SYK P43405 1/20 0.35
ATR Q13535 1/20 0.34
AURKA O14965 2/20 0.33
RPS6KB1 P23443 2/20 0.33
NR2E1 Q9Y466 1/20 0.33
CCR9 P51686 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CYP3A4 P08684 2/20 0.33
FAAH O00519 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
KDR P35968 1/20 0.33
WNT3A P56704 1/20 0.33
AGPAT2 O15120 1/20 0.32
NQO2 P16083 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780029 0.85 CNR1 (0.39) KCNK3KCNK9CNR1PLCG1SYK
SCHEMBL4793442 0.84 HPGDS (0.45) KCNK3KCNK9CNR1PLCG1
SCHEMBL3931030 0.83 KCNK3 (0.43) KCNK3KCNK9CNR1AURKARPS6KB1
SCHEMBL3929384 0.79 HPGDS (0.43) KCNK3KCNK9CNR1PLCG1
SCHEMBL3929850 0.76 HPGDS (0.45) KCNK3KCNK9
SCHEMBL3939593 0.76 KCNK3 (0.46) KCNK3KCNK9CNR1NR2E1CCR9
SCHEMBL4780033 0.74 KCNK3 (0.39) KCNK3KCNK9CNR1AURKAHDAC4
SCHEMBL4796842 0.73 HPGDS (0.46) PLCG1
SCHEMBL4795668 0.73 HPGDS (0.46) PLCG1
SCHEMBL3933505 0.72 PIP4K2A (0.52) KCNK3KCNK9CCR9CYP3A4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090093479-A1 ANTI-CANCER AGENTS AND USES THEREOF LOCUS PHARMACEUTICALS, INC. (US) 2009-04-09 US disclosed
US-7504401-B2 Anti-cancer agents and uses thereof LOCUS PHARMACEUTICALS, INC. (US) 2009-03-17 US disclosed
US-20080280891-A1 Anti-cancer agents and uses thereof LOCUS PHARMACEUTICALS, INC. (US) 2008-11-13 US disclosed
WO-2008008059-A1 ANTI-CANCER AGENTS ANS USES THEREOF LOCUS PHARMACEUTICALS, INC. (US) 2008-01-17 WO disclosed
US-20060270686-A1 Anti-cancer agents and uses thereof LOCUS PHARMACEUTICALS, INC. 2006-11-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090093479-A1 ANTI-CANCER AGENTS AND USES THEREOF H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, MCL1, CBR3 KCNK3 1783/4885KCNK9 3501/4885CNR1 196/4885
US-20060270686-A1 Anti-cancer agents and uses thereof H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, MCL1, CBR3 KCNK3 1797/4885KCNK9 3554/4885CNR1 233/4885
US-20080280891-A1 Anti-cancer agents and uses thereof NR2E3, RB1, CBR3 KCNK3 1938/4885KCNK9 3675/4885CNR1 202/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.