SCHEMBL3940689

SCHEMBL3940689

O=C(Nc1ccccc1C(=O)c1ccccc1)C(=O)Nc1ccccc1C(=O)c1ccccc1

nearest known ligand 0.69

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.67
KMT2A Q03164 3/20 0.59
AKR1C3 P42330 1/20 0.55
TRPA1 O75762 1/20 0.53
MAPT P10636 3/20 0.52
GAA P10253 2/20 0.52
MEN1 O00255 2/20 0.51
PKM P14618 1/20 0.51
BDKRB1 P46663 2/20 0.49
LMNA P02545 1/20 0.49
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
USP2 O75604 1/20 0.47
KEAP1 Q14145 1/20 0.47
NFE2L2 Q16236 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
TP53 P04637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14397784 0.92 ALDH1A1 (0.63) ALDH1A1KMT2AAKR1C3TRPA1MAPT
SCHEMBL27580953 0.89 ALDH1A1 (0.59) ALDH1A1KMT2AAKR1C3TRPA1MAPT
SCHEMBL4678464 0.88 ALDH1A1 (0.67) ALDH1A1KMT2AAKR1C3MAPTGAA
SCHEMBL83108 0.86 ALDH1A1 (0.65) ALDH1A1KMT2AAKR1C3MAPTGAA
SCHEMBL819016 0.86 MAPT (0.66) ALDH1A1KMT2AMAPTMEN1PKM
SCHEMBL10725281 0.86 ALDH1A1 (0.56) ALDH1A1KMT2AAKR1C3TRPA1MAPT
SCHEMBL12683508 0.85 ALDH1A1 (0.55) ALDH1A1KMT2AAKR1C3TRPA1MAPT
SCHEMBL28228800 0.85 ALDH1A1 (0.63) ALDH1A1KMT2AAKR1C3MAPTGAA
SCHEMBL2047090 0.85 CYP2C19 (0.66) ALDH1A1KMT2AAKR1C3MAPTBDKRB1
SCHEMBL8174226 0.83 KMT2A (0.62) ALDH1A1KMT2AAKR1C3MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218004-B1 5-METHYL INDIRUBIN FOR USE IN THE TREATMENT OF HUMAN SOLID TUMORS FIEBIG HEINZ HERBERT (DE) 2009-04-08 EP disclosed
US-6664285-B1 Administering for treatment of human solid tumors and metastasis thereof EISENBRAND GERHARD (DE) 2003-12-16 US disclosed