SCHEMBL3943602

SCHEMBL3943602

COC[C@@H](C)NC(=O)c1[nH]c2ccc(NS(=O)(=O)c3ccc(C(C)(C)C)cc3)cc2c1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.50
SERPINE1 P05121 1/20 0.48
CA1 P00915 3/20 0.45
CA2 P00918 3/20 0.45
CA12 O43570 1/20 0.45
CA4 P22748 1/20 0.45
CA6 P23280 1/20 0.45
CA5A P35218 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45
CA14 Q9ULX7 1/20 0.45
CA5B Q9Y2D0 1/20 0.45
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
POLB P06746 2/20 0.43
ALDH1A1 P00352 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3952380 1.00 BRD4 (0.50) BRD4SERPINE1CA1CA2CA12
SCHEMBL3947589 1.00 BRD4 (0.50) BRD4SERPINE1CA1CA2CA12
SCHEMBL3953037 0.91 BRD4 (0.52) BRD4SERPINE1CA1CA2CA12
SCHEMBL3946187 0.89 BRD4 (0.52) BRD4SERPINE1CA1CA2CA12
SCHEMBL3952994 0.87 BRD4 (0.49) BRD4SERPINE1CA1CA2KMT2A
SCHEMBL3951354 0.87 BRD4 (0.49) BRD4SERPINE1CA1CA2KMT2A
SCHEMBL3944739 0.87 BRD4 (0.49) BRD4SERPINE1CA1CA2KMT2A
SCHEMBL5149516 0.86 CA1 (0.49) BRD4SERPINE1CA1CA2CA12
SCHEMBL3951651 0.85 HTR6 (0.47) BRD4SERPINE1CA1CA2CA12
SCHEMBL3950163 0.85 BRD4 (0.51) BRD4SERPINE1CA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1802572-B1 INDOL DERIVATIVES AS INHIBITORS OF SOLUBLE ADENYLYL CYCLASE BAYER SCHERING PHARMA AG (DE) 2009-04-22 EP claimed