SCHEMBL3943702

SCHEMBL3943702

O=C(Nc1ccc(Cl)c(C(=O)Nc2cccnc2)c1)c1cc(F)cc(C2CC2)c1

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 12/20 0.70
BRAF P15056 3/20 0.54
CYP11B2 P19099 2/20 0.50
NAMPT P43490 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3934404 0.89 CSF1R (0.83) CSF1RBRAFCYP11B2L3MBTL1
SCHEMBL1276598 0.89 BRAF (0.70) CSF1RBRAF
SCHEMBL1276906 0.87 CSF1R (0.74) CSF1RBRAFCYP11B2
SCHEMBL3934893 0.86 CSF1R (0.85) CSF1RBRAFCYP11B2NAMPTL3MBTL1
SCHEMBL3938937 0.84 CSF1R (0.86) CSF1RBRAF
SCHEMBL3934183 0.83 CSF1R (1.00) CSF1RBRAFL3MBTL1
SCHEMBL3929957 0.82 CSF1R (0.78) CSF1RBRAF
SCHEMBL3932168 0.80 CSF1R (0.60) CSF1RBRAF
SCHEMBL3932812 0.78 CSF1R (1.00) CSF1RBRAFCYP11B2
SCHEMBL3936075 0.78 CSF1R (1.00) CSF1RBRAFCYP11B2NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1831198-B1 PYRIDINE CARBOXAMIDE DERIVATIVES FOR USE AS ANTICANCER AGENTS ASTRAZENECA AB (SE) 2009-04-08 EP disclosed
CN-101128454-A Pyridine carboxamide derivatives for use as anticancer agents ASTRAZENECA AB (SE) 2008-02-20 CN disclosed