SCHEMBL3944545

SCHEMBL3944545

[CH2]CC(C)(O)C(Cc1ccccc1)C(N)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.46
ALPI P09923 1/20 0.42
PKM P14618 1/20 0.42
PTGS1 P23219 1/20 0.42
XIAP P98170 1/20 0.42
SLC7A5 Q01650 1/20 0.42
CYP1A2 P05177 1/20 0.41
POLB P06746 2/20 0.40
ALDH1A1 P00352 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
SRR Q9GZT4 2/20 0.39
SLC1A3 P43003 1/20 0.39
SLC1A2 P43004 1/20 0.39
SLC1A1 P43005 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
ALPL P05186 1/20 0.38
ALPG P10696 1/20 0.38
KDM4E B2RXH2 1/20 0.38
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14591098 0.82 EPHX1 (0.53) EPHX1ALPIPKMPTGS1XIAP
SCHEMBL15426320 0.82 EPHX1 (0.53) EPHX1ALPIPKMPTGS1XIAP
SCHEMBL6648151 0.75 EPHX1 (0.53) EPHX1ALPIPKMPTGS1XIAP
SCHEMBL20394045 0.71 CYP1A2 (0.52) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL13248648 0.71 ALPI (0.44) EPHX1ALPIPKMPTGS1XIAP
SCHEMBL27503896 0.71 EPHX1 (0.49) EPHX1ALPIPKMPTGS1XIAP
SCHEMBL66965 0.71 CYP1A2 (0.55) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL15426321 0.71 CYP1A2 (0.55) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL19787829 0.71 TRPA1 (0.45) EPHX1ALPIPKMPTGS1XIAP
SCHEMBL12650596 0.69 ALPI (0.50) ALPIPKMPTGS1XIAPSLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2046755-A2 PYRAZOLES AS GLUCOKINASE ACTIVATORS F. Hoffmann-Roche AG (CH) 2009-04-15 EP disclosed
WO-2008012227-A2 PYRAZOLES AS GLUCOKINASE ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2008-01-31 WO disclosed