SCHEMBL3948699

SCHEMBL3948699

O=Cc1ccc2c(c1)NC=CS2

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 1/20 0.34
PTGS2 P35354 1/20 0.34
RAB9A P51151 1/20 0.34
CYP2A6 P11509 4/20 0.33
KIF11 P52732 2/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ALDH1A3 P47895 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11277664 0.69 NOX1 (0.43) ALDH1A1KDM4EPTGS2RAB9ACYP2A6
SCHEMBL5515460 0.68 ALDH1A1 (0.42) ALDH1A1KDM4EPTGS2RAB9ACYP2A6
SCHEMBL27648588 0.66 CYP2A6 (0.38) ALDH1A1KDM4EPTGS2RAB9ACYP2A6
SCHEMBL31083349 0.63 ALDH1A1 (0.50) ALDH1A1KDM4EPTGS2RAB9ACYP2A6
SCHEMBL31083569 0.63 ALDH1A1 (0.50) ALDH1A1KDM4EPTGS2RAB9ACYP2A6
SCHEMBL11272621 0.63 NOX1 (0.59) ALDH1A1PTGS2RAB9ATSHRHSD17B10
SCHEMBL3054155 0.63 ALDH1A1 (0.49) ALDH1A1KDM4EPTGS2RAB9ACYP2A6
SCHEMBL27476532 0.63 ALDH1A1 (0.33) ALDH1A1KDM4EPTGS2RAB9ACYP2A6
SCHEMBL6440717 0.63 ALDH1A1 (0.37) ALDH1A1KDM4EPTGS2RAB9ACYP2A6
SCHEMBL622422 0.62 HTT (0.56) ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009020457-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-02-12 WO disclosed
EP-2010532-A1 TRYCLIC NITROGEN CONTAINING COMPOUNDS AND THEIR USE AS ANTIBACTERIALS Glaxo Group Limited (GB) 2009-01-07 EP disclosed
WO-2007122258-A1 TRYCLIC NITROGEN CONTAINING COMPOUNDS AND THEIR USE AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2007-11-01 WO disclosed