SCHEMBL3953232

SCHEMBL3953232

Nc1cncc(C(Br)Br)n1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 1/20 0.44
GRM4 Q14833 1/20 0.33
HSP90AA1 P07900 1/20 0.32
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31226557 0.74 CDK2 (0.43) CDK2GRM4HSP90AA1NOS3NOS1
SCHEMBL31226663 0.74 CDK2 (0.43) CDK2GRM4HSP90AA1NOS3NOS1
SCHEMBL31226309 0.74 CDK2 (0.43) CDK2GRM4HSP90AA1NOS3NOS1
SCHEMBL1604498 0.73
Hydrochloric Acid SCHEMBL31108166 0.70
Hydrochloric Acid SCHEMBL31108165 0.70
SCHEMBL22426961 0.70 CDK2 (0.39) CDK2GRM4NOS3NOS1NOS2
SCHEMBL24796831 0.69 CDK2 (0.38) CDK2
SCHEMBL20692815 0.69 CDK2 (0.42) CDK2
SCHEMBL24016972 0.69 CDK2 (0.38) CDK2NOS3NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2078016-A2 HETEROARYL COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH Signal Pharmaceuticals LLC (US) 2009-07-15 EP disclosed
WO-2008051493-A2 HETEROARYL COMPOUNDS, COMPOSITIONS THEREOF, AND THEIR USE AS PROTEIN KINASE INHIBITORS SIGNAL PHARMACEUTICALS, LLC (US) 2008-05-02 WO disclosed