SCHEMBL3956211

SCHEMBL3956211

CCOC(=O)CSc1nc(-c2cc(OC)c(C#N)cc2Cl)c2c(C#N)cn(COCC[Si](C)(C)C)c2n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 7/20 0.47
HSP90AA1 P07900 3/20 0.46
KCNH2 Q12809 3/20 0.43
PIM1 P11309 1/20 0.36
ALDH1A1 P00352 4/20 0.35
KDM4E B2RXH2 3/20 0.35
MAPT P10636 3/20 0.35
RAB9A P51151 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 2/20 0.35
ABCB1 P08183 1/20 0.35
USP2 O75604 1/20 0.35
NFKB1 P19838 1/20 0.35
CASP1 P29466 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35
HSD17B10 Q99714 1/20 0.35
HPGD P15428 3/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4134884 0.93 HSP90AB1 (0.50) HSP90AB1HSP90AA1KCNH2PIM1ALDH1A1
SCHEMBL2567338 0.92 HSP90AB1 (0.47) HSP90AB1HSP90AA1KCNH2PIM1ALDH1A1
SCHEMBL4064357 0.91 HSP90AB1 (0.48) HSP90AB1HSP90AA1KCNH2TDP1L3MBTL1
SCHEMBL3955735 0.87 HSP90AA1 (0.62) HSP90AB1HSP90AA1KCNH2SMN1; SMN2
SCHEMBL2566599 0.86 KCNH2 (0.43) HSP90AB1HSP90AA1KCNH2
SCHEMBL2564620 0.85 HSP90AB1 (0.55) HSP90AB1HSP90AA1KCNH2PIM1
SCHEMBL13798712 0.84 KCNH2 (0.62) HSP90AB1HSP90AA1KCNH2
SCHEMBL3961239 0.84 HSP90AA1 (0.56) HSP90AB1HSP90AA1KCNH2SMN1; SMN2GAA
SCHEMBL3961424 0.84 HSP90AB1 (0.42) HSP90AB1HSP90AA1KCNH2ALDH1A1RAB9A
SCHEMBL3956701 0.83 HSP90AB1 (0.48) HSP90AB1HSP90AA1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009030871-A1 PYRROLOPYRIMIDINE DERIVATIVES HAVING HSP90 INHIBITORY ACTIVITY VERNALIS R & D LTD (GB) 2009-03-12 WO disclosed