SCHEMBL4134884

SCHEMBL4134884

CCOC(=O)CSc1nc(-c2cc(O)c(OC)cc2Cl)c2c(C#N)cn(COCC[Si](C)(C)C)c2n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AB1 P08238 7/20 0.50
HSP90AA1 P07900 3/20 0.49
KCNH2 Q12809 3/20 0.37
PIM1 P11309 1/20 0.36
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 2/20 0.34
MAPT P10636 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
RAB9A P51151 2/20 0.34
ABCB1 P08183 1/20 0.34
TNF P01375 1/20 0.34
NPC1 O15118 1/20 0.34
USP2 O75604 1/20 0.34
NFKB1 P19838 1/20 0.34
CASP1 P29466 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
HSD17B10 Q99714 1/20 0.34
HPGD P15428 2/20 0.34
L3MBTL1 Q9Y468 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3956211 0.93 HSP90AB1 (0.47) HSP90AB1HSP90AA1KCNH2PIM1ALDH1A1
SCHEMBL3961239 0.91 HSP90AA1 (0.56) HSP90AB1HSP90AA1KCNH2SMN1; SMN2
SCHEMBL2567338 0.91 HSP90AB1 (0.47) HSP90AB1HSP90AA1KCNH2PIM1ALDH1A1
SCHEMBL3961248 0.90 HSP90AB1 (0.56) HSP90AB1HSP90AA1KCNH2LMNA
SCHEMBL3955015 0.86 HSP90AB1 (0.53) HSP90AB1HSP90AA1KCNH2ALDH1A1KDM4E
SCHEMBL3955735 0.86 HSP90AA1 (0.62) HSP90AB1HSP90AA1KCNH2SMN1; SMN2
SCHEMBL2569133 0.85 HSP90AB1 (0.46) HSP90AB1HSP90AA1KCNH2
SCHEMBL4064357 0.84 HSP90AB1 (0.48) HSP90AB1HSP90AA1KCNH2L3MBTL1
SCHEMBL2567033 0.84 HSP90AB1 (0.44) HSP90AB1HSP90AA1KCNH2PIM1ALDH1A1
SCHEMBL2564620 0.84 HSP90AB1 (0.55) HSP90AB1HSP90AA1KCNH2PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090163490-A1 Pyrrolopyrimidine Derivatives Used As HSP90 Inhibitors VERNALIS (R&D) LTD. (GB) 2009-06-25 US disclosed
US-20090163490-A1 Pyrrolopyrimidine Derivatives Used As HSP90 Inhibitors VERNALIS (R&D) LTD. (GB) 2009-06-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090163490-A1 Pyrrolopyrimidine Derivatives Used As HSP90 Inhibitors HSP90AA1, HSP90AB1, RAF1 HSP90AB1 2/4885HSP90AA1 1/4885KCNH2 2202/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.