SCHEMBL3957262

SCHEMBL3957262

CN[C@H](C/C=C/c1cncc(OC)c1)COP(=O)(O)O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.47
CHRNA4 P43681 3/20 0.47
ROCK2 O75116 1/20 0.40
MAP4K4 O95819 1/20 0.40
PRKACA P17612 1/20 0.40
ROCK1 Q13464 1/20 0.40
DYRK1A Q13627 1/20 0.40
NTRK3 Q16288 1/20 0.40
PKN2 Q16513 1/20 0.40
CLK4 Q9HAZ1 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
STK17A Q9UEE5 1/20 0.40
CHRNB4 P30926 1/20 0.38
CHRNA3 P32297 1/20 0.38
CHRNA7 P36544 1/20 0.38
LPAR3 Q9UBY5 4/20 0.32
LPAR1 Q92633 3/20 0.32
GRIK1 P39086 1/20 0.32
GRIK2 Q13002 1/20 0.32
PLA2G4A P47712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2329000 0.89 CHRNB2 (0.63) CHRNB2CHRNA4CHRNB4CHRNA3CHRNA7
SCHEMBL3952130 0.82 CHRNB2 (0.47) CHRNB2CHRNA4ROCK2MAP4K4PRKACA
SCHEMBL3961184 0.82 CHRNB2 (0.47) CHRNB2CHRNA4ROCK2MAP4K4PRKACA
Phosphoric Acid SCHEMBL3957257 0.81 CHRNB2 (0.67) CHRNB2CHRNA4ROCK2MAP4K4PRKACA
SCHEMBL3959982 0.77 CHRNB2 (0.43) CHRNB2CHRNA4ROCK2MAP4K4PRKACA
SCHEMBL3954681 0.77 CHRNB2 (0.42) CHRNB2CHRNA4ROCK2MAP4K4PRKACA
SCHEMBL621495 0.76 CHRNB2 (0.78) CHRNB2CHRNA4ROCK2MAP4K4PRKACA
SCHEMBL617913 0.76 CHRNB2 (0.78) CHRNB2CHRNA4ROCK2MAP4K4PRKACA
SCHEMBL620296 0.76 CHRNB2 (0.78) CHRNB2CHRNA4ROCK2MAP4K4PRKACA
SCHEMBL620297 0.76 CHRNB2 (0.78) CHRNB2CHRNA4ROCK2MAP4K4PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009018367-A2 NOVEL SALT FORMS OF (2S)-(4E)-N-METHYL-5-[3-(5-METHOXYPYRIDIN)YL]-4-PENTEN-2-AMINE TARGACEPT, INC. (US) 2009-02-05 WO claimed
WO-2009018367-A2 NOVEL SALT FORMS OF (2S)-(4E)-N-METHYL-5-[3-(5-METHOXYPYRIDIN)YL]-4-PENTEN-2-AMINE TARGACEPT, INC. (US) 2009-02-05 WO disclosed