SCHEMBL3958975

SCHEMBL3958975

COc1ccc2c(c1)CCN(C1CCN(C(=O)CN)CC1)C(=O)N2

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 15/20 0.43
ACHE P22303 1/20 0.43
CBX7 O95931 1/20 0.41
CDYL2 Q8N8U2 1/20 0.41
CDYL Q9Y232 1/20 0.41
RAMP1 O60894 3/20 0.41
ALDH1A1 P00352 2/20 0.40
GLA P06280 1/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
DPP4 P27487 1/20 0.40
USP2 O75604 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3964416 0.88 ALDH1A1 (0.41) CALCRLACHECBX7CDYL2CDYL
SCHEMBL4079721 0.87 PDE3B (0.41) CALCRLRAMP1DPP4
SCHEMBL1700431 0.84 PDE3B (0.46) ALDH1A1
SCHEMBL3963894 0.83 PDE3B (0.40)
SCHEMBL30178252 0.83 CBX7 (0.41) CALCRLACHECBX7CDYL2CDYL
SCHEMBL30178610 0.83 ALDH1A1 (0.51) ALDH1A1
SCHEMBL3960086 0.82 CALCRL (0.55) CALCRLRAMP1
SCHEMBL5374732 0.82 CALCRL (0.41) CALCRLACHECBX7CDYL2CDYL
SCHEMBL13907937 0.82 ALDH1A1 (0.38) CALCRLCBX7CDYL2CDYLRAMP1
SCHEMBL4079724 0.81 PDE3B (0.40) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034029-A2 1-SUBSTITUTED 4-HETEROCYCLYLPIPERIDINES FOR USE AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-19 WO disclosed