SCHEMBL3961573

SCHEMBL3961573

CCOC(=O)c1cncc(C)c1Cl

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.48
TSHR P16473 1/20 0.47
MEN1 O00255 2/20 0.47
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
ALDH1A1 P00352 5/20 0.45
CASP1 P29466 1/20 0.43
NPC1 O15118 2/20 0.43
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
CYP4F2 P78329 1/20 0.42
CYP4A11 Q02928 1/20 0.42
BAZ2B Q9UIF8 1/20 0.42
BAZ2A Q9UIF9 1/20 0.42
METTL3 Q86U44 1/20 0.42
POLB P06746 1/20 0.41
RAB9A P51151 1/20 0.41
HSD17B10 Q99714 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2567016 0.91 TSHR (0.52) KMT2ATSHRMEN1CYP2C9CYP2C19
SCHEMBL1521876 0.86 KMT2A (0.48) KMT2ATSHRMEN1CYP2C9CYP2C19
SCHEMBL2567248 0.83 KMT2A (0.46) KMT2ATSHRMEN1CYP2C9CYP2C19
SCHEMBL3828694 0.83 ATM (0.35) KMT2AMEN1CYP2C9CYP2C19ALDH1A1
SCHEMBL21558450 0.82 ATM (0.44) TSHRALDH1A1NPC1LMNASMN1; SMN2
SCHEMBL21866062 0.81 KMT2A (0.44) KMT2ATSHRMEN1CYP2C9CYP2C19
SCHEMBL2649492 0.81 HSP90AA1 (0.46) KMT2ATSHRMEN1CYP2C9CYP2C19
SCHEMBL5267090 0.80 KDM4E (0.50) KMT2ATSHRMEN1ALDH1A1POLB
SCHEMBL3913326 0.79 ALDH1A1 (0.53) KMT2ATSHRMEN1CYP2C9CYP2C19
SCHEMBL9590155 0.79 KMT2A (0.42) KMT2ATSHRMEN1CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079690-A2 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES Actelion Pharmaceuticals Ltd. (CH) 2009-07-22 EP disclosed
WO-2008038251-A2 3-AZA-BICYCLO[3.1.0]HEXANE DERIVATIVES ACTELION PHARMACEUTICALS LTD (CH) 2008-04-03 WO disclosed