Clioquinol

Clioquinol

SCHEMBL3967

Oc1c(I)cc(Cl)c2cccnc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 1.00
LMNA P02545 5/20 1.00
MEN1 O00255 5/20 1.00
HTT P42858 5/20 1.00
KMT2A Q03164 5/20 1.00
SMN1; SMN2 Q16637 5/20 1.00
TDP1 Q9NUW8 5/20 1.00
HSP90AA1 P07900 5/20 1.00
MAPT P10636 5/20 1.00
METAP2 P50579 5/20 1.00
ALDH1A1 P00352 4/20 1.00
TP53 P04637 3/20 1.00
ALOX15 P16050 3/20 1.00
SLC6A2 P23975 3/20 1.00
MMP14 P50281 3/20 1.00
OPRK1 P41145 3/20 1.00
ALOX12 P18054 3/20 1.00
USP2 O75604 2/20 1.00
CYP3A4 P08684 2/20 1.00
HPGD P15428 2/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Clioquinol SCHEMBL29370380 1.00 KDM4E (1.00) KDM4ELMNAMEN1HTTKMT2A
Clioquinol SCHEMBL30592904 1.00 KDM4E (1.00) KDM4ELMNAMEN1HTTKMT2A
Clioquinol SCHEMBL11749381 1.00 KDM4E (1.00) KDM4ELMNAMEN1HTTKMT2A
Clioquinol SCHEMBL27671588 0.98 KDM4E (0.97) KDM4ELMNAMEN1HTTKMT2A
Clioquinol SCHEMBL18985133 0.98 KDM4E (0.97) KDM4ELMNAMEN1HTTKMT2A
Clioquinol SCHEMBL28198183 0.98 KDM4E (0.97) KDM4ELMNAMEN1HTTKMT2A
Clioquinol SCHEMBL28531298 0.98 KDM4E (0.97) KDM4ELMNAMEN1HTTKMT2A
Clioquinol SCHEMBL28529781 0.98 KDM4E (0.97) KDM4ELMNAMEN1HTTKMT2A
Clioquinol SCHEMBL28524321 0.98 KDM4E (0.97) KDM4ELMNAMEN1HTTKMT2A
Clioquinol SCHEMBL9339556 0.98 KDM4E (0.97) KDM4ELMNAMEN1HTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 13819 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026106952-A1 METHODS FOR TREATING CONGENITAL DISORDERS OF GLYCOSYLATION CDG CARE (US) 2026-05-21 WO claimed
EP-4255391-B1 LUMINOL FOR USE IN THE TREATMENT OF SEQUELAE OF A SARS-COV-2 INFECTION METRIOPHARM AG (CH) 2026-05-06 EP claimed
EP-4719412-A1 2,8-DIHYDROXYQUINOLINE GLUCURONIDE DERIVATIVES WITH ENHANCED PROPERTIES FOR USE AS ANTICANCER, ANTIVIRAL, ANTIMICROBIAL, AND OTHER THERAPEUTIC APPLICATIONS Westol, LLC (US) 2026-04-08 EP claimed
US-12590963-B2 Anti-cancer treatment of preselected subjects and screening methods to identify susceptible subjects TUDAG TU DRESDEN AKTIENGESELLSCHAFT (DE) 2026-03-31 US claimed
EP-4640714-A2 METHODS FOR ASSESSING RISK OF DEVELOPING A VIRAL DISEASE USING A GENETIC TEST PML Screening, LLC (US) 2025-10-29 EP claimed
EP-4632063-A2 COPPER LOSS MITIGATION GENENTECH, INC. (US) 2025-10-15 EP claimed
EP-3824059-B1 CLEANING COMPOSITION WITH CORROSION INHIBITOR ENTEGRIS INC (US) 2025-09-17 EP claimed
US-20250248940-A1 Biopolymer Formulations for Drug Delivery 11584022 CANADA INC. (CA) 2025-08-07 US claimed
US-20250248988-A1 COMBINATION USES OF NITROXOLINE AND ITS ANALOGUES WITH CHEMOTHERAPIES AND IMMUNOTHERAPIES IN THE TREATMENT OF CANCERS JIANGSU YAHONG MEDITECH CO., LTD. (CN) 2025-08-07 US claimed
EP-4136211-B1 COPPER LOSS MITIGATION GENENTECH INC (US) 2025-07-09 EP claimed
EP-0046270-B1 NOVEL DERIVATIVES OF BIO-AFFECTING PHENOLIC COMPOUNDS AND PHARMACEUTICAL COMPOSITION CONTAINING THEM INTERx RESEARCH CORPORATION (US) 1986-05-21 EP claimed
US-4520099-A CONTAINING AN HYDROXYQUINOLINE AS AN ANTIFOGGING AGENT FUJI PHOTO FILM CO., LTD. (JP) 1985-05-28 US claimed
US-4485091-A HYDROGEN PEROXIDE, OIL IN WATER EMULSION QUINODERM LIMITED (GB) 1984-11-27 US claimed
EP-0035856-B1 PHARMACEUTICAL AND DIETARY COMPOSITIONS EFAMOL LIMITED (GB) 1984-07-04 EP claimed
EP-0098577-A2 Drugs for treating diarrhea caused by infection HOECHST AKTIENGESELLSCHAFT (DE) 1984-01-18 EP claimed
EP-0096457-A1 Indium complexes of substituted 8-hydroxy-quinolines, pharmaceutical compositions containing them and their use as antibacterial agents NATIONAL RESEARCH DEVELOPMENT CORPORATION (GB) 1983-12-21 EP claimed
EP-0046270-A1 Novel derivatives of bio-affecting phenolic compounds and pharmaceutical composition containing them INTERx RESEARCH CORPORATION (US) 1982-02-24 EP claimed
EP-0037175-A1 Pharmaceutical compositions EFAMOL LIMITED (GB) 1981-10-07 EP claimed
EP-0035856-A2 Pharmaceutical and dietary compositions EFAMOL LIMITED (GB) 1981-09-16 EP claimed
WO-1980000791-A1 B-GLUCURONIDASE ACTIVITY AND/OR PH-DEPENDENT PHARMACEUTICALS AND THEIR METHODS OF PRODUCTION AND USE FOR SELECTIVE TREATMENT OF DISEASES SCHWIMMER A (US) 1980-05-01 WO claimed