SCHEMBL3969296

SCHEMBL3969296

N#Cc1ccc2sc(-c3nc(Nc4ccc(OCCN5CCCC5)cc4)nc4[nH]ccc34)cc2c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 3/20 0.40
AXL P30530 3/20 0.39
CDK1 P06493 1/20 0.39
KDR P35968 1/20 0.39
BRAF P15056 1/20 0.39
PRKCQ Q04759 3/20 0.39
CACNA1B Q00975 2/20 0.39
INSR P06213 1/20 0.39
TBK1 Q9UHD2 1/20 0.38
PRKCD Q05655 2/20 0.38
CACNA1H O95180 1/20 0.38
SRC P12931 1/20 0.38
HRH3 Q9Y5N1 2/20 0.38
LTA4H P09960 1/20 0.38
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
JAK2 O60674 1/20 0.37
JAK3 P52333 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13883460 0.94 BACE1 (0.40) BACE1AXLCDK1KDRBRAF
SCHEMBL13883619 0.89 AXL (0.43) BACE1AXLKDRINSRSRC
SCHEMBL3966481 0.88 BACE1 (0.48) BACE1AXLKDRINSRSRC
SCHEMBL3967611 0.85 AXL (0.45) AXLKDRPRKCQINSRPRKCD
SCHEMBL3967636 0.83 AXL (0.55) AXLCDK1KDRBRAFINSR
SCHEMBL3969198 0.82 WEE1 (0.39) BACE1AXLCDK1KDRSRC
SCHEMBL13883588 0.82 HDAC1 (0.43) HRH3JAK2JAK3
SCHEMBL13883580 0.81 AXL (0.46) BACE1AXLKDRINSRSRC
SCHEMBL3971213 0.81 TTK (0.56) JAK2JAK3
SCHEMBL3964683 0.80 AXL (0.48) BACE1AXLCDK1KDRINSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009049028-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USE AS JANUS KINASE MODULATORS TARGEGEN INC. (US) 2009-04-16 WO disclosed
WO-2009049028-A1 PYRROLOPYRIMIDINE COMPOUNDS AND THEIR USE AS JANUS KINASE MODULATORS TARGEGEN INC. (US) 2009-04-16 WO disclosed