SCHEMBL3970914

SCHEMBL3970914

CCOc1cc(CN(c2ccc(C#N)cn2)C2CCNCC2)ccc1O

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 3/20 0.41
SLC6A2 P23975 8/20 0.40
SLC6A4 P31645 8/20 0.40
SLC6A3 Q01959 6/20 0.40
CYP19A1 P11511 1/20 0.38
JAK2 O60674 2/20 0.37
JAK3 P52333 2/20 0.37
KDM1A O60341 1/20 0.36
MAPKAPK2 P49137 1/20 0.35
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35
TSHR P16473 2/20 0.35
HTR6 P50406 1/20 0.35
KCNH2 Q12809 1/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
HPGD P15428 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3972421 0.90 SLC6A2 (0.41) IKBKBSLC6A2SLC6A4SLC6A3JAK2
SCHEMBL3973911 0.89 SLC6A2 (0.40) IKBKBSLC6A2SLC6A4SLC6A3CYP19A1
SCHEMBL3976469 0.89 SLC6A2 (0.40) IKBKBSLC6A2SLC6A4SLC6A3JAK2
SCHEMBL3972485 0.89 SLC6A2 (0.40) IKBKBSLC6A2SLC6A4SLC6A3JAK2
SCHEMBL3972502 0.87 SLC6A2 (0.39) IKBKBSLC6A2SLC6A4SLC6A3JAK2
SCHEMBL3973888 0.87 IKBKB (0.40) IKBKBSLC6A2SLC6A4SLC6A3JAK2
SCHEMBL3973733 0.87 SLC6A2 (0.39) IKBKBSLC6A2SLC6A4SLC6A3JAK2
SCHEMBL3972380 0.87 SLC6A2 (0.39) IKBKBSLC6A2SLC6A4SLC6A3JAK2
SCHEMBL3973372 0.84 RXRA (0.41) SLC6A2SLC6A4SLC6A3KDM4EALDH1A1
SCHEMBL3977612 0.83 SLC6A2 (0.37) IKBKBSLC6A2SLC6A4SLC6A3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP claimed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO claimed
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP disclosed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO disclosed