SCHEMBL3971263

SCHEMBL3971263

COc1cccc(C#CC2(O)CCCC(NC(C)=O)C2)c1.COc1cccc(C#CC2(O)CCCC(NC(C)=O)C2)c1

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 14/20 0.58
MTNR1A P48039 2/20 0.42
MTNR1B P49286 2/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL990085 1.00 GRM5 (0.58) GRM5MTNR1AMTNR1BNPC1RAB9A
SCHEMBL3627130 0.92 GRM5 (0.58) GRM5NPC1RAB9ASMN1; SMN2CYP1A2
SCHEMBL990697 0.87 GRM5 (0.53) GRM5NPC1RAB9ASMN1; SMN2CYP1A2
SCHEMBL990047 0.87 GRM5 (0.53) GRM5SMN1; SMN2CYP1A2CYP3A4CYP2C19
SCHEMBL990750 0.86 GRM5 (0.56) GRM5
SCHEMBL990045 0.85 GRM5 (0.54) GRM5CYP2C19
SCHEMBL990721 0.80 GRM5 (0.56) GRM5
SCHEMBL990246 0.79 GRM5 (0.58) GRM5
SCHEMBL14119620 0.78 GRM5 (0.54) GRM5
SCHEMBL5744089 0.78 GRM5 (0.52) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009047303-A2 METABOTROPIC GLUTAMATE RECEPTOR MODULATORS FOR THE TREATMENT OF PERVASIVE DEVELOPMENTAL DISORDER NOVARTIS AG (CH) 2009-04-16 WO disclosed