SCHEMBL3973709

SCHEMBL3973709

CCCCCCCNc1cc(C(=O)O)ccc1C(N)=O

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 5/20 0.56
CISD1 Q9NZ45 6/20 0.50
PLK1 P53350 4/20 0.50
XDH P47989 1/20 0.46
TP53 P04637 1/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3141041 0.99 HCAR3 (0.57) HCAR3CISD1PLK1XDHTSHR
SCHEMBL2427920 0.94 HCAR3 (0.56) HCAR3CISD1PLK1TSHR
SCHEMBL22097725 0.90 HCAR3 (0.60) HCAR3CISD1PLK1XDH
SCHEMBL2425639 0.89 HCAR3 (0.55) HCAR3CISD1
SCHEMBL3975310 0.87 HCAR3 (0.46) HCAR3CISD1PLK1TSHR
SCHEMBL3980340 0.85 PTGER4 (0.56) HCAR3PLK1
SCHEMBL22097708 0.84 HCAR3 (0.60) HCAR3CISD1PLK1TSHR
SCHEMBL27972972 0.83 KDM6B (0.55) HCAR3CISD1PLK1TSHR
SCHEMBL2432061 0.83 MAPT (0.62) HCAR3
SCHEMBL18272540 0.83 PTGER4 (0.56) HCAR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074120-A1 TROPANE COMPOUNDS Exelixis, Inc. (US) 2009-07-01 EP disclosed
WO-2009055077-A1 TROPANE COMPOUNDS EXELIXIS, INC. (US) 2009-04-30 WO disclosed