SCHEMBL3975447

SCHEMBL3975447

NC(=O)c1ccc(-c2ccccc2)c(F)c1OCCBr

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 2/20 0.44
ALOX5AP P20292 3/20 0.37
FEN1 P39748 3/20 0.37
IKBKB O14920 3/20 0.36
PLA2G2A P14555 3/20 0.36
PLA2G10 O15496 2/20 0.36
BRD4 O60885 1/20 0.35
KDM4E B2RXH2 1/20 0.35
PDK2 Q15119 1/20 0.34
PARP10 Q53GL7 1/20 0.34
CHUK O15111 1/20 0.34
IKBKE Q14164 1/20 0.34
PKMYT1 Q99640 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3981622 0.86 BCAT2 (0.44) BCAT2ALOX5APFEN1IKBKBPLA2G2A
SCHEMBL3974955 0.85 BCAT2 (0.43) BCAT2IKBKBPLA2G2APLA2G10BRD4
SCHEMBL3975515 0.83 BCAT2 (0.54) BCAT2IKBKBPLA2G2APLA2G10KDM4E
SCHEMBL23573105 0.76 BCAT2 (0.58) BCAT2ALOX5APFEN1IKBKBPLA2G2A
SCHEMBL3979295 0.72 BCAT2 (0.43) BCAT2IKBKBPLA2G2APLA2G10BRD4
SCHEMBL3974889 0.71 MKNK1 (0.47) KDM4EPARP10HTTSMN1; SMN2
SCHEMBL30841448 0.70 BCAT2 (0.69) BCAT2IKBKBKDM4EPDK2HTT
SCHEMBL3973836 0.69 BCAT2 (0.54) BCAT2IKBKBKDM4EHTTSMN1; SMN2
SCHEMBL18816701 0.69 BCAT2 (0.53) BCAT2IKBKBBRD4KDM4EPARP10
SCHEMBL27674225 0.69 BCAT2 (0.49) BCAT2IKBKBPLA2G2APLA2G10BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054383-A2 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS AT OPIOID RECEPTORS SmithKline Beecham Corporation (US) 2009-05-06 EP disclosed
WO-2008021849-A2 NOVEL COMPOUNDS AS ANTAGONISTS OR INVERSE AGONISTS AT OPIOID RECEPTORS SMITHKLINE BEECHAM CORPORATION (US) 2008-02-21 WO disclosed