SCHEMBL3975634

SCHEMBL3975634

COc1ccc2c(c1)CCC(c1ccccc1)=C2C(O)c1ccc(OCCN2CCCC2)cc1

nearest known ligand 0.72

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
EBP Q15125 1/20 0.72
SIGMAR1 Q99720 1/20 0.72
LTA4H P09960 5/20 0.57
ESR1 P03372 7/20 0.54
ESR2 Q92731 6/20 0.54
HRH3 Q9Y5N1 2/20 0.47
PTPN1 P18031 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7521111 0.99 EBP (0.70) EBPSIGMAR1LTA4HESR1ESR2
SCHEMBL13897747 0.94 EBP (0.66) EBPSIGMAR1LTA4HESR1ESR2
SCHEMBL7105837 0.94 EBP (0.62) EBPSIGMAR1LTA4HESR1ESR2
SCHEMBL7524285 0.94 EBP (0.65) EBPSIGMAR1LTA4HESR1ESR2
SCHEMBL13897766 0.94 EBP (0.65) EBPSIGMAR1LTA4HESR1ESR2
SCHEMBL7109994 0.93 EBP (0.61) EBPSIGMAR1LTA4HESR1ESR2
SCHEMBL7108683 0.90 EBP (0.59) EBPSIGMAR1LTA4HESR1ESR2
SCHEMBL3869661 0.89 EBP (0.58) EBPSIGMAR1ESR1ESR2HRH3
SCHEMBL3861283 0.89 EBP (0.58) EBPSIGMAR1LTA4HESR1ESR2
SCHEMBL7109917 0.88 EBP (0.56) EBPSIGMAR1LTA4HHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7501441-B1 Naphthyl compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 2009-03-10 US disclosed
US-7501441-B1 Naphthyl compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 2009-03-10 US disclosed
US-7501441-B1 Naphthyl compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY (US) 2009-03-10 US disclosed
US-6437137-B1 REDUCING (NAPHTHALEN-1-YL)(4-(2-(1-PIPERDINYL)ETHOXY) PHENYL)METHANONE WITH A REDUCING AGENT IN THE PRESENCE OF A SOLVENT, HEATING TO REFLUX; FORMING (NAPHTHALEN-1-YL)(4-(2-(1-PIPERDINYL)ETHOXY)PHENYL)METHANE ELI LILLY AND COMPANY 2002-08-20 US disclosed
EP-0702961-B1 Compositions for minimizing the uterotrophic effect of tamoxifen and its analogs LILLY CO ELI (US) 2002-07-24 EP disclosed
US-6410564-B1 Naphthyl compounds, intermediates, processes, compositions, and methods ELI LILLY AND COMPANY 2002-06-25 US disclosed
US-5658931-A ADMINISTERING A MIXTURE OF ANTIESTROGENS ELI LILLY AND COMPANY (US) 1997-08-19 US disclosed
US-5554628-A A 1-(4-ALKOXYPHENYL-)NAPHTHALENE COMPOUND ELI LILLY AND COMPANY (US) 1996-09-10 US disclosed
WO-1996009052-A1 A METHOD FOR INHIBITING MAMMALIAN BREAST CARCINOMA WITH TAMOXIFEN, AND ANALOGS THEREOF, AND CERTAIN NAPHTHYL COMPOUNDS ELI LILLY AND COMPANY (US) 1996-03-28 WO disclosed
WO-1996009039-A1 NAPHTHYL COMPOUNDS, INTERMEDIATES, PROCESSES, COMPOSITIONS, AND METHODS ELI LILLY AND COMPANY (US) 1996-03-28 WO disclosed
EP-0702962-A2 Preparations for inhibiting mammalian breast carcinoma with tamoxifen and analogs thereof, and certain naphthyl compounds ELI LILLY AND COMPANY (US) 1996-03-27 EP disclosed
EP-0702961-A2 Compositions for minimizing the uterotrophic effect of tamoxifen and its analogs ELI LILLY AND COMPANY (US) 1996-03-27 EP disclosed
EP-0703228-A1 Naphthyl compounds, intermediates, processes, compositions involving them ELI LILLY AND COMPANY (US) 1996-03-27 EP disclosed
US-5484796-A Naphthyl compounds, intermediates, processes, compositions, and method of inhibiting aortal smooth muscle cell proliferation ELI LILLY AND COMPANY (US) 1996-01-16 US disclosed
US-5484795-A Naphthyl compounds, intermediates, processes, compositions, and method of inhibiting restenosis ELI LILLY AND COMPANY (US) 1996-01-16 US disclosed
US-5484797-A Naphthly compounds, intermediates, processes, compositions, and method for inhibiting endometrosis ELI LILLY AND COMPANY (US) 1996-01-16 US disclosed