SCHEMBL3976004

SCHEMBL3976004

O=c1c(I)n[nH]c2ccccc12

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.61
KDM4E B2RXH2 7/20 0.58
ALDH1A1 P00352 3/20 0.58
NPC1 O15118 1/20 0.58
TP53 P04637 1/20 0.58
RAB9A P51151 1/20 0.58
GAA P10253 3/20 0.50
PDPK1 O15530 1/20 0.50
CYP3A4 P08684 1/20 0.50
POLB P06746 1/20 0.48
HPGD P15428 2/20 0.48
LMNA P02545 1/20 0.48
GLA P06280 1/20 0.48
HTT P42858 1/20 0.48
ATM Q13315 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
IDO1 P14902 3/20 0.47
ALPL P05186 1/20 0.47
TTK P33981 1/20 0.47
MAPK10 P53779 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL516645 0.83 KDM4E (0.58) CYP1A2KDM4EALDH1A1NPC1TP53
SCHEMBL30163026 0.83 KDM4E (0.58) CYP1A2KDM4EALDH1A1NPC1TP53
SCHEMBL1023212 0.78 CYP1A2 (0.63) CYP1A2KDM4EALDH1A1NPC1TP53
SCHEMBL9041896 0.76 CYP1A2 (0.61) CYP1A2KDM4EALDH1A1NPC1TP53
SCHEMBL6480580 0.76 CYP1A2 (1.00) CYP1A2KDM4EALDH1A1NPC1TP53
SCHEMBL9042255 0.76 KDM4E (0.73) CYP1A2KDM4EALDH1A1NPC1TP53
SCHEMBL25357544 0.74 JAK2 (0.56) CYP1A2PDPK1IDO1LRRK2CDK2
SCHEMBL31010860 0.74 MAP2K4 (0.50) KDM4EALDH1A1GAAGLAHTT
SCHEMBL30310978 0.74 ITK (0.45) CYP1A2NPC1POLBMAP2K4CHEK1
SCHEMBL21591507 0.73 CYP1A2 (0.58) CYP1A2KDM4EALDH1A1NPC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009053799-A1 NOVEL CANNABINOID RECEPTOR LIGANDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND PROCESS FOR THEIR PREPARATION GLENMARK PHARMACEUTICALS, S.A. (US) 2009-04-30 WO disclosed
WO-2009053799-A1 NOVEL CANNABINOID RECEPTOR LIGANDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND PROCESS FOR THEIR PREPARATION GLENMARK PHARMACEUTICALS, S.A. (US) 2009-04-30 WO disclosed