SCHEMBL3976467

SCHEMBL3976467

CCOc1cc(CN2CCC(N(c3ccc(C(F)(F)F)cn3)N(c3ccc(C(F)(F)F)cn3)C3CCN(Cc4ccc(OC)c(OCC)c4)CC3)CC2)ccc1Cl

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.51
ALDH1A1 P00352 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
RAB9A P51151 1/20 0.46
SSTR5 P35346 14/20 0.44
HRH1 P35367 4/20 0.44
SSTR1 P30872 1/20 0.44
HTR2B P41595 2/20 0.42
DRD4 P21917 1/20 0.42
OPRD1 P41143 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3971377 0.86 SSTR5 (0.41) KDM4EALDH1A1NPSR1SSTR5HRH1
SCHEMBL3977762 0.81 SSTR5 (0.52) KDM4EALDH1A1SSTR5HRH1HTR2B
SCHEMBL3977776 0.79 SSTR5 (0.50) KDM4EALDH1A1SSTR5HRH1HTR2B
SCHEMBL3972896 0.79 SSTR5 (0.43) KDM4EALDH1A1NPSR1SSTR5
SCHEMBL4000512 0.78 SSTR5 (0.46) KDM4EALDH1A1NPSR1SSTR5HRH1
SCHEMBL2418270 0.78 SSTR5 (0.56) SSTR5HRH1SSTR1HTR2B
SCHEMBL2415066 0.78 SSTR5 (0.56) KDM4EALDH1A1NPSR1RAB9ASSTR5
SCHEMBL3939333 0.78 SSTR5 (0.47) KDM4EALDH1A1NPSR1SSTR5HRH1
SCHEMBL3997966 0.76 SSTR5 (0.44) KDM4EALDH1A1NPSR1RAB9ASSTR5
SCHEMBL3971809 0.73 SSTR5 (0.52) SSTR5HRH1SSTR1HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2054385-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. Hoffmann-Roche AG (CH) 2009-05-06 EP disclosed
WO-2008019967-A2 PHENYL, PYRIDINE AND QUINOLINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2008-02-21 WO disclosed