SCHEMBL3977441

SCHEMBL3977441

COc1cccc(CCNC(=O)c2ccc(N3C4CC[C@H]3CC(NC(=O)c3cccc(OC)c3C)C4)nc2)c1

nearest known ligand 0.77

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 14/20 0.77
HSP90AB1 P08238 14/20 0.77
ROCK2 O75116 1/20 0.47
ROCK1 Q13464 1/20 0.47
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2425134 0.93 HSP90AA1 (0.85) HSP90AA1HSP90AB1ROCK2ROCK1
SCHEMBL2425132 0.93 HSP90AA1 (0.85) HSP90AA1HSP90AB1ROCK2ROCK1
SCHEMBL3980048 0.92 HSP90AA1 (0.87) HSP90AA1HSP90AB1RAB9A
SCHEMBL2426782 0.92 HSP90AA1 (0.75) HSP90AA1HSP90AB1
SCHEMBL2426780 0.92 HSP90AA1 (0.75) HSP90AA1HSP90AB1
SCHEMBL2429263 0.90 HSP90AA1 (0.77) HSP90AA1HSP90AB1RAB9A
SCHEMBL2429266 0.90 HSP90AA1 (0.77) HSP90AA1HSP90AB1RAB9A
SCHEMBL2427717 0.89 HSP90AA1 (0.84) HSP90AA1HSP90AB1
SCHEMBL2427718 0.89 HSP90AA1 (0.84) HSP90AA1HSP90AB1
SCHEMBL2428574 0.89 HSP90AA1 (0.76) HSP90AA1HSP90AB1ROCK2ROCK1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074120-A1 TROPANE COMPOUNDS Exelixis, Inc. (US) 2009-07-01 EP disclosed
WO-2009055077-A1 TROPANE COMPOUNDS EXELIXIS, INC. (US) 2009-04-30 WO disclosed