SCHEMBL3979898

SCHEMBL3979898

CCOP(=O)(CCN(C1CCNCC1)S(=O)(=O)c1ccc(Nc2nccc(Nc3ccc(F)cc3)n2)cc1)OCC

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
LMNA P02545 1/20 0.42
MAPT P10636 1/20 0.42
ALOX12 P18054 1/20 0.42
MAPK1 P28482 1/20 0.42
RAB9A P51151 1/20 0.42
KMT2A Q03164 1/20 0.42
SYK P43405 1/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
KCNH2 Q12809 2/20 0.39
SLC6A3 Q01959 1/20 0.39
KDR P35968 2/20 0.38
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
CDK2 P24941 3/20 0.37
CHRNA7 P36544 1/20 0.36
CDK4 P11802 1/20 0.36
CCNE1 P24864 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4441619 0.93 IKBKB (0.42) MEN1NPC1LMNAMAPTALOX12
SCHEMBL4883643 0.85 MEN1 (0.47) MEN1NPC1LMNAMAPTALOX12
SCHEMBL4622257 0.85 MEN1 (0.48) MEN1NPC1LMNAMAPTALOX12
SCHEMBL4622719 0.85 MEN1 (0.46) MEN1NPC1LMNAMAPTALOX12
Hydrochloric Acid SCHEMBL4885375 0.84 MEN1 (0.47) MEN1NPC1LMNAMAPTALOX12
SCHEMBL14020157 0.84 MEN1 (0.49) MEN1NPC1LMNAMAPTALOX12
Hydrochloric Acid SCHEMBL4883215 0.84 MEN1 (0.45) MEN1NPC1LMNAMAPTALOX12
SCHEMBL14020199 0.84 DRD2 (0.40) MEN1NPC1LMNAMAPTALOX12
SCHEMBL14020209 0.84 DRD2 (0.39) MEN1NPC1LMNAMAPTALOX12
Hydrochloric Acid SCHEMBL4882044 0.83 MEN1 (0.48) MEN1NPC1LMNAMAPTALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009056693-A1 NOVEL DERIVATIVES OF N, N'- 2, 4-DIANILINOPYRIMIDINES, PREPARATION THEREOF AS MEDICAMENTS PHARMACEUTICAL COMPOSITIONS AND IN PARTICULAR AS IKK INHIBITORS SANOFI-AVENTIS (FR) 2009-05-07 WO disclosed