Bicarbonate

Bicarbonate

SCHEMBL3980487

COc1ccc(C2(C#N)CCN(C3CC3)CC2)cc1OCC1CC1.O=C(O)O

nearest known ligand 0.69

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 20/20 0.69
PDE4A P27815 19/20 0.69
PDE4C Q08493 19/20 0.69
PDE4D Q08499 19/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3160937 0.86 PDE4B (0.81) PDE4BPDE4APDE4CPDE4D
SCHEMBL3160359 0.86 PDE4B (0.69) PDE4BPDE4APDE4CPDE4D
SCHEMBL6546903 0.84 PDE4B (0.76) PDE4BPDE4APDE4CPDE4D
SCHEMBL6546476 0.84 PDE4B (0.76) PDE4BPDE4APDE4CPDE4D
SCHEMBL6546469 0.84 PDE4B (0.76) PDE4BPDE4APDE4CPDE4D
Bicarbonate SCHEMBL3982339 0.83 PDE4A (0.71) PDE4BPDE4APDE4CPDE4D
Bicarbonate SCHEMBL3981807 0.83 PDE4A (0.74) PDE4BPDE4APDE4CPDE4D
SCHEMBL6820943 0.83 PDE4B (0.66) PDE4BPDE4APDE4CPDE4D
SCHEMBL6545648 0.83 PDE4B (0.66) PDE4BPDE4APDE4CPDE4D
SCHEMBL6545650 0.83 PDE4B (0.66) PDE4BPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1308440-B1 PIPERIDINE DERIVATIVES AND DRUGS CONTAINING THESE DERIVATIVES AS THE ACTIVE INGREDIENT ONO PHARMACEUTICAL CO (JP) 2009-05-06 EP claimed