SCHEMBL3982575

SCHEMBL3982575

O=C(NCc1ccc2cc(C(=O)O)sc2c1)c1ccccc1

nearest known ligand 0.83

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 11/20 0.83
SENP5 Q96HI0 1/20 0.58
SENP2 Q9HC62 1/20 0.58
SENP1 Q9P0U3 1/20 0.58
ERCC1 P07992 1/20 0.55
ERCC4 Q92889 1/20 0.55
BCL2L1 Q07817 1/20 0.51
NR1H4 Q96RI1 1/20 0.51
HDAC2 Q92769 2/20 0.50
HDAC3 O15379 1/20 0.50
NCOR2 Q9Y618 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
PPARG P37231 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1885089 0.91 HDAC1 (1.00) HDAC1SENP5SENP2SENP1HDAC2
SCHEMBL4075809 0.86 HDAC1 (0.63) HDAC1NR1H4CYP2C9CYP2C19PPARG
SCHEMBL3568348 0.83 HDAC2 (0.72) HDAC1SENP5SENP2SENP1HDAC2
SCHEMBL3565538 0.81 HDAC1 (0.74) HDAC1ERCC1ERCC4BCL2L1HDAC2
SCHEMBL3570753 0.80 HDAC1 (0.57) HDAC1SENP5SENP2SENP1BCL2L1
SCHEMBL1884493 0.79 HDAC1 (0.78) HDAC1HDAC2HDAC3HDAC6CYP2C19
SCHEMBL1889752 0.79 HDAC1 (0.78) HDAC1HDAC2HDAC3NCOR2HDAC6
SCHEMBL4255241 0.78 HDAC1 (0.82) HDAC1BCL2L1
SCHEMBL8291123 0.78 HDAC1 (1.00) HDAC1HDAC2HDAC3HDAC6CYP2C9
SCHEMBL1890070 0.78 HDAC1 (0.81) HDAC1HDAC2HDAC3HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1677731-A4 THIOPHENE AND BENZOTHIOPHENE HYDROXAMIC ACID DERIVATIVES ATON PHARMA INC (US) 2009-05-06 EP disclosed
EP-1677731-A2 THIOPHENE AND BENZOTHIOPHENE HYDROXAMIC ACID DERIVATIVES Aton Pharma, Inc. (US) 2006-07-12 EP disclosed
WO-2005034880-A2 THIOPHENE AND BENZOTHIOPHENE HYDROXAMIC ACID DERIVATIVES ATON PHARMA, INC. (US) 2005-04-21 WO disclosed