SCHEMBL3982633

SCHEMBL3982633

CCNc1nc2c(C(=O)O)cccc2o1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 4/20 0.56
ELANE P08246 2/20 0.43
TOP2A P11388 2/20 0.43
IDO1 P14902 1/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
ALDH1A1 P00352 1/20 0.40
CA12 O43570 3/20 0.38
CA9 Q16790 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
MAPT P10636 1/20 0.37
PKM P14618 1/20 0.37
MAPK1 P28482 1/20 0.37
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
TP53 P04637 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CA2 P00918 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1005317 0.86 HTR3A (0.54) HTR3AELANETOP2AALDH1A1SMN1; SMN2
SCHEMBL1005664 0.84 HTR3A (0.54) HTR3AELANETOP2AIDO1MAOA
SCHEMBL1008152 0.83 TOP2A (0.45) HTR3ATOP2AIDO1MAOAMAOB
SCHEMBL1003671 0.82 HTR3A (0.41) HTR3AELANETOP2AIDO1MAOA
SCHEMBL1006835 0.82 HTR3A (0.41) HTR3ATOP2AIDO1MAOAMAOB
Hydrochloric Acid SCHEMBL1004329 0.82 HTR3A (0.41) HTR3ATOP2AIDO1MAOAMAOB
Hydrochloric Acid SCHEMBL1007973 0.82 HTR3A (0.41) HTR3AELANETOP2AIDO1MAOA
SCHEMBL1006463 0.81 HTR3A (0.43) HTR3AELANETOP2AIDO1MAOA
SCHEMBL27776060 0.79 KDM4E (0.48) TOP2AALDH1A1SMN1; SMN2MAPTMAPK1
SCHEMBL19298146 0.78 IDO1 (0.44) HTR3AELANETOP2AIDO1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101528225-B 2-aminobenzoxazole carboxamides as 5HT3 modulators ALBANY MOLECULAR RES INC 2013-07-17 CN disclosed
CN-101528225-A 2-aminobenzoxazole carboxamides as 5HT3 modulators AMR TECHNOLOGY INC (US) 2009-09-09 CN disclosed
EP-2061460-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS Albany Molecular Research, Inc. (US) 2009-05-27 EP disclosed
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed