SCHEMBL3984271

SCHEMBL3984271

Cc1ccc2oc(N3CCOCC3CC(C)C)nc2c1C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 9/20 0.53
MDM2 Q00987 2/20 0.37
KCNH2 Q12809 1/20 0.33
LRRK2 Q5S007 1/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
GRM2 Q14416 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
HCRTR1 O43613 3/20 0.31
HCRTR2 O43614 3/20 0.31
LMNA P02545 1/20 0.31
HTT P42858 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
FKBP1A P62942 1/20 0.31
CYP3A4 P08684 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1006857 1.00 HTR3A (0.53) HTR3AMDM2KCNH2LRRK2ALDH1A1
SCHEMBL1004321 0.89 HTR3A (0.51) HTR3AKCNH2NPC1RAB9A
SCHEMBL1005156 0.89 HTR3A (0.51) HTR3AKCNH2NPC1RAB9A
SCHEMBL1004322 0.89 HTR3A (0.51) HTR3AKCNH2NPC1RAB9A
SCHEMBL1007977 0.87 HTR3A (0.52) HTR3AKCNH2ALDH1A1L3MBTL1NPC1
SCHEMBL1007978 0.87 HTR3A (0.52) HTR3AKCNH2ALDH1A1L3MBTL1NPC1
SCHEMBL1006355 0.86 HTR3A (0.52) HTR3AKCNH2ALDH1A1L3MBTL1FKBP1A
SCHEMBL1006356 0.86 HTR3A (0.52) HTR3AKCNH2ALDH1A1L3MBTL1FKBP1A
SCHEMBL1006363 0.86 HTR3A (0.52) HTR3AKCNH2ALDH1A1L3MBTL1FKBP1A
SCHEMBL1005780 0.84 HTR3A (0.49) HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061460-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS Albany Molecular Research, Inc. (US) 2009-05-27 EP disclosed
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed