SCHEMBL3984568

SCHEMBL3984568

CN1C2CCCC1CC(NC(=O)c1cccc3oc(NC4CN(C(C)(C)C)C4)nc13)C2

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 20/20 0.67
KCNH2 Q12809 4/20 0.67
CYP2C19 P33261 1/20 0.60
CYP3A4 P08684 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1005319 0.92 HTR3A (0.75) HTR3AKCNH2CYP2C19CYP3A4
Hydrochloric Acid SCHEMBL1005350 0.91 HTR3A (0.74) HTR3AKCNH2CYP2C19CYP3A4
SCHEMBL1006331 0.89 HTR3A (0.71) HTR3AKCNH2CYP2C19CYP3A4
SCHEMBL1004897 0.88 HTR3A (0.61) HTR3AKCNH2CYP2C19CYP3A4
Hydrochloric Acid SCHEMBL1006445 0.88 HTR3A (0.70) HTR3AKCNH2CYP2C19CYP3A4
SCHEMBL12928076 0.87 HTR3A (0.72) HTR3AKCNH2CYP2C19CYP3A4
Hydrochloric Acid SCHEMBL1006451 0.86 HTR3A (0.71) HTR3AKCNH2CYP2C19CYP3A4
SCHEMBL1004167 0.86 HTR3A (0.75) HTR3AKCNH2CYP2C19CYP3A4
Hydrochloric Acid SCHEMBL1005603 0.85 HTR3A (0.74) HTR3AKCNH2CYP2C19CYP3A4
SCHEMBL8222503 0.83 HTR3A (0.71) HTR3AKCNH2CYP2C19CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061460-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS Albany Molecular Research, Inc. (US) 2009-05-27 EP disclosed
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed