SCHEMBL3984595

SCHEMBL3984595

COC(=O)c1cccc2oc(C3CNc4ccccc4N3)nc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 2/20 0.47
HSD17B10 Q99714 2/20 0.39
ALOX5 P09917 1/20 0.37
HTR3A P46098 2/20 0.37
KCNH2 Q12809 2/20 0.37
PKN1 Q16512 1/20 0.37
PKN2 Q16513 1/20 0.37
RIPK1 Q13546 1/20 0.37
KDM4E B2RXH2 5/20 0.37
ALDH1A1 P00352 2/20 0.37
HPGD P15428 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 1/20 0.35
NPC1 O15118 4/20 0.35
RAB9A P51151 4/20 0.35
KMT2A Q03164 3/20 0.34
ATM Q13315 3/20 0.34
MAPT P10636 2/20 0.34
GAA P10253 2/20 0.34
MEN1 O00255 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3984630 0.87 MAOB (0.38) TOP2AALOX5HTR3AKCNH2KDM4E
SCHEMBL4308323 0.74 TOP2A (0.51) TOP2AHSD17B10HTR3AKCNH2PKN1
SCHEMBL1007865 0.72 TOP2A (0.43) TOP2AHSD17B10HTR3AKCNH2PKN1
SCHEMBL14721812 0.70 GAA (0.42) ALOX5KDM4EALDH1A1SMN1; SMN2RAB9A
SCHEMBL1398896 0.70 TOP2A (0.59) TOP2AHSD17B10PKN1PKN2RIPK1
SCHEMBL4311643 0.69 HTR3A (0.48) TOP2AHSD17B10HTR3AKCNH2RIPK1
SCHEMBL1003473 0.69 TOP2A (0.45) TOP2AHSD17B10ALOX5HTR3AKCNH2
SCHEMBL1005898 0.69 TOP2A (0.57) TOP2AHSD17B10PKN1PKN2RIPK1
SCHEMBL1121666 0.69 TOP2A (0.57) TOP2AHSD17B10PKN1PKN2RIPK1
SCHEMBL1004337 0.69 TOP2A (0.57) TOP2AHSD17B10HTR3APKN1PKN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061460-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS Albany Molecular Research, Inc. (US) 2009-05-27 EP disclosed
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed