SCHEMBL3984928

SCHEMBL3984928

CC1CN(C(C)(C)C)CCN1c1nc2c(C(=O)NC3CC4CCN3CC4)cccc2o1

nearest known ligand 0.50

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 20/20 0.50
KCNH2 Q12809 3/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1006362 0.86 HTR3A (0.47) HTR3AKCNH2CYP2C19
Hydrochloric Acid SCHEMBL1005553 0.82 HTR3A (0.69) HTR3AKCNH2CYP2C19
SCHEMBL1004466 0.81 HTR3A (0.66) HTR3AKCNH2CYP2C19
SCHEMBL1005720 0.81 HTR3A (0.67) HTR3AKCNH2CYP2C19
Hydrochloric Acid SCHEMBL1005562 0.80 HTR3A (0.66) HTR3AKCNH2CYP2C19
Hydrochloric Acid SCHEMBL1004299 0.80 HTR3A (0.65) HTR3AKCNH2CYP2C19
SCHEMBL1004856 0.79 HTR3A (0.46) HTR3AKCNH2CYP2C19
SCHEMBL1006786 0.79 HTR3A (0.51) HTR3AKCNH2CYP2C19
SCHEMBL1005533 0.78 HTR3A (0.57) HTR3AKCNH2CYP2C19
Hydrochloric Acid SCHEMBL1005891 0.78 HTR3A (0.45) HTR3AKCNH2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061460-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS Albany Molecular Research, Inc. (US) 2009-05-27 EP disclosed
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed