SCHEMBL3984963

SCHEMBL3984963

COC(=O)c1cccc2oc(N3C(C)CN(C(C)=O)CC3C)nc12

nearest known ligand 0.52

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 17/20 0.52
KCNH2 Q12809 4/20 0.48
CYP2C19 P33261 1/20 0.48
TOP2A P11388 2/20 0.45
HCRTR1 O43613 1/20 0.37
HCRTR2 O43614 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1005918 1.00 HTR3A (0.52) HTR3AKCNH2CYP2C19TOP2AHCRTR1
SCHEMBL3990444 0.89 HTR3A (0.49) HTR3AKCNH2CYP2C19TOP2A
SCHEMBL1005434 0.89 HTR3A (0.49) HTR3AKCNH2CYP2C19TOP2A
SCHEMBL1006097 0.88 HTR3A (0.51) HTR3AKCNH2CYP2C19TOP2A
SCHEMBL3988561 0.88 HTR3A (0.51) HTR3AKCNH2CYP2C19TOP2A
SCHEMBL1004469 0.87 HTR3A (0.48) HTR3AKCNH2CYP2C19TOP2AHCRTR2
SCHEMBL1004355 0.87 HTR3A (0.48) HTR3AKCNH2CYP2C19TOP2AHCRTR2
SCHEMBL3984149 0.87 HTR3A (0.50) HTR3AKCNH2CYP2C19TOP2A
SCHEMBL1005157 0.87 HTR3A (0.48) HTR3AKCNH2CYP2C19TOP2AHCRTR2
SCHEMBL1005158 0.87 HTR3A (0.48) HTR3AKCNH2CYP2C19TOP2AHCRTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061460-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS Albany Molecular Research, Inc. (US) 2009-05-27 EP disclosed
WO-2008019372-A2 2-AMINOBENZOXAZOLE CARBOXAMIDES AS 5HT3 MODULATORS ALBANY MOLECULAR RESEARCH, INC. (US) 2008-02-14 WO disclosed