SCHEMBL3986970

SCHEMBL3986970

c1ccc(-c2cc[nH]c2-c2ccc[nH]2)nc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.49
KDM4E B2RXH2 5/20 0.43
LMNA P02545 3/20 0.43
CCR1 P32246 2/20 0.43
CCR5 P51681 2/20 0.43
CCR8 P51685 2/20 0.43
CYP1A2 P05177 1/20 0.43
POLB P06746 1/20 0.43
METAP1 P53582 1/20 0.43
BLM P54132 1/20 0.43
HIF1A Q16665 1/20 0.43
DOHH Q9BU89 1/20 0.43
P4HTM Q9NXG6 1/20 0.43
KDM4C Q9H3R0 1/20 0.40
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
TP53 P04637 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
ALOX15 P16050 2/20 0.38
HTT P42858 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL404747 0.83 PRKCI (0.56) PRKCIKDM4ELMNACCR1CCR5
SCHEMBL28264205 0.82 PRKCI (0.54) PRKCIKDM4ELMNACCR1CCR5
SCHEMBL439769 0.81 KDM4E (0.54) PRKCIKDM4ELMNACCR1CCR5
SCHEMBL29529148 0.81 KDM4E (0.54) PRKCIKDM4ELMNACCR1CCR5
SCHEMBL27768754 0.80 KDM4E (0.52) PRKCIKDM4ELMNACCR1CCR5
Pyridine SCHEMBL28181012 0.75 KDM4C (0.49) PRKCIKDM4ELMNACCR1CCR5
SCHEMBL21578438 0.75 KDM4E (0.46) PRKCIKDM4ELMNACCR1CCR5
SCHEMBL28504411 0.75 IDO1 (0.43) PRKCIKDM4ELMNACCR1CCR5
SCHEMBL18204056 0.74 KDM4E (0.64) PRKCIKDM4ELMNACCR1CCR5
SCHEMBL3992598 0.73 CCR1 (0.47) CCR1CCR8TGFBR1MAPK14METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2061785-A2 LINEAR PYRIDAZINE AND PYRROLE COMPOUNDS, PROCESSES FOR OBTAINING THEM AND USES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2009-05-27 EP claimed
WO-2008012441-A2 LINEAR PYRIDAZINE AND PYRROLE COMPOUNDS, PROCESSES FOR OBTAINING THEM AND USES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S.) (FR) 2008-01-31 WO claimed
EP-2061785-A2 LINEAR PYRIDAZINE AND PYRROLE COMPOUNDS, PROCESSES FOR OBTAINING THEM AND USES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2009-05-27 EP disclosed
WO-2008012441-A2 LINEAR PYRIDAZINE AND PYRROLE COMPOUNDS, PROCESSES FOR OBTAINING THEM AND USES CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S.) (FR) 2008-01-31 WO disclosed