SCHEMBL398925

SCHEMBL398925

O=C(O)c1cccnc1N1CCSCC1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.65
MYC P01106 1/20 0.53
KDM4E B2RXH2 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
CYP3A4 P08684 2/20 0.46
TSHR P16473 2/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPT P10636 1/20 0.46
ALOX15 P16050 1/20 0.46
BLM P54132 1/20 0.46
AGER Q15109 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MEN1 O00255 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
CHIA Q9BZP6 1/20 0.46
HSD17B10 Q99714 1/20 0.45
NAPRT Q6XQN6 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3309889 0.85 KMT2A (0.70) KMT2AMYCKDM4ETDP1CYP3A4
SCHEMBL15294735 0.85 KMT2A (0.70) KMT2AMYCKDM4ETDP1CYP3A4
SCHEMBL30477850 0.85 KMT2A (0.70) KMT2AMYCKDM4ETDP1CYP3A4
SCHEMBL17746092 0.84 KMT2A (0.68) KMT2AMYCKDM4ETDP1CYP3A4
SCHEMBL31057148 0.84 KMT2A (0.68) KMT2AMYCKDM4ETDP1CYP3A4
SCHEMBL11399275 0.84 KMT2A (0.68) KMT2AMYCKDM4ETDP1CYP3A4
SCHEMBL7234041 0.83 KMT2A (0.67) KMT2AMYCKDM4ETDP1CYP3A4
SCHEMBL394318 0.82 OPRK1 (0.54) KMT2AKDM4ETDP1CYP3A4MAPT
SCHEMBL7243430 0.81 KMT2A (0.65) KMT2AMYCKDM4ETDP1TSHR
SCHEMBL593819 0.81 KMT2A (0.69) KMT2AMYCKDM4ETDP1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408745-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2012-01-25 EP disclosed