SCHEMBL3989395

SCHEMBL3989395

CC(=O)Cc1ccc(-c2ccccc2)c(-c2ccc(C(F)(F)F)cc2)n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.51
PSEN1 P49768 1/20 0.44
PSEN2 P49810 1/20 0.44
APH1B Q8WW43 1/20 0.44
NCSTN Q92542 1/20 0.44
APH1A Q96BI3 1/20 0.44
PSENEN Q9NZ42 1/20 0.44
PTGDR2 Q9Y5Y4 2/20 0.44
DHODH Q02127 2/20 0.42
S1PR3 Q99500 7/20 0.42
KIF11 P52732 1/20 0.41
DPP4 P27487 1/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
APP P05067 1/20 0.40
PDE2A O00408 1/20 0.39
RXRA P19793 1/20 0.39
RXRB P28702 1/20 0.39
RXRG P48443 1/20 0.39
CYP2C8 P10632 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3996379 1.00 BACE1 (0.51) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL3991979 0.88 S1PR3 (0.48) PTGDR2S1PR3LMNA
SCHEMBL2833946 0.81 BACE1 (0.51) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL3995229 0.80 KIF11 (0.44) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL2834553 0.78 BACE1 (0.45) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL2833627 0.78 BACE1 (0.45) BACE1PSEN1PSEN2APH1BNCSTN
SCHEMBL2837655 0.75 BACE1 (0.48) BACE1DHODHKIF11APP
SCHEMBL2832416 0.75 BACE1 (0.48) BACE1DHODHKIF11APP
SCHEMBL2830992 0.75 DHODH (0.54) BACE1DHODHLMNAHTT
SCHEMBL2831678 0.75 DHODH (0.54) BACE1DHODHLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2064183-A2 HETEROAROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR AGONIST BIOLOGICAL ACTIVITY Allergan, Inc. (US) 2009-06-03 EP disclosed
WO-2008030838-A2 HETEROAROMATIC COMPOUNDS HAVING SPHINGOSINE-1-PHOSPHATE (S1P) RECEPTOR AGONIST BIOLOGICAL ACTIVITY ALLERGAN, INC. (US) 2008-03-13 WO disclosed