SCHEMBL3990678

SCHEMBL3990678

CN(Cc1nc2ccccc2n1C[C@H]1CCCN(C(NC(=O)OC(C)(C)C)NC(=O)OC(C)(C)C)C1)[C@@H]1CCCc2cccnc21

nearest known ligand 0.73

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 18/20 0.73
CYP3A4 P08684 1/20 0.39
SCN9A Q15858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3993664 1.00 CXCR4 (0.73) CXCR4CYP3A4SCN9A
SCHEMBL4935802 0.87 CXCR4 (0.70) CXCR4
SCHEMBL4938545 0.85 CXCR4 (1.00) CXCR4
SCHEMBL4287996 0.85 CXCR4 (1.00) CXCR4
SCHEMBL4938546 0.85 CXCR4 (1.00) CXCR4
SCHEMBL4933539 0.85 CXCR4 (1.00) CXCR4
SCHEMBL3998366 0.84 CXCR4 (0.66) CXCR4
SCHEMBL4125051 0.84 CXCR4 (0.61) CXCR4
SCHEMBL4935750 0.83 CXCR4 (0.65) CXCR4
SCHEMBL4940055 0.83 CXCR4 (0.64) CXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778231-A4 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2009-06-03 EP disclosed
EP-1778231-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-05-02 EP disclosed
WO-2006020415-A1 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2006-02-23 WO disclosed