SCHEMBL4006486

SCHEMBL4006486

CCc1ncnc2[nH]cc(Br)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 2/20 0.39
TNNI3K Q59H18 2/20 0.39
MAPK1 P28482 2/20 0.36
CHEK1 O14757 2/20 0.36
IRAK4 Q9NWZ3 3/20 0.35
PLK4 O00444 2/20 0.35
ROCK2 O75116 2/20 0.35
PRKD3 O94806 2/20 0.35
MAP4K4 O95819 2/20 0.35
CDK1 P06493 2/20 0.35
FES P07332 2/20 0.35
ROS1 P08922 2/20 0.35
FGFR1 P11362 2/20 0.35
PHKG2 P15735 2/20 0.35
PRKACA P17612 2/20 0.35
RPS6KB1 P23443 2/20 0.35
CDK2 P24941 2/20 0.35
MARK3 P27448 2/20 0.35
FLT4 P35916 2/20 0.35
FLT3 P36888 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14330947 0.80 AKT1 (0.44) BRAFTNNI3KCHEK1IRAK4PLK4
SCHEMBL24392119 0.79 NOTUM (0.47) BRAFTNNI3KMAPK1CHEK1IRAK4
SCHEMBL7885565 0.76 MAPK1 (0.39) BRAFTNNI3KMAPK1CHEK1IRAK4
SCHEMBL19306619 0.76 BRAF (0.41) BRAFTNNI3KMAPK1CHEK1IRAK4
SCHEMBL17401156 0.75 MAP3K7 (0.56) IRAK4ROCK2CHUKROCK1CDC42BPA
SCHEMBL868756 0.73 RET (0.41) BRAFTNNI3KMAPK1CHEK1IRAK4
SCHEMBL22096107 0.72 STK3 (0.61) BRAFTNNI3KMAPK1CHEK1IRAK4
SCHEMBL154600 0.72 CHEK1 (0.61) BRAFTNNI3KMAPK1CHEK1DYRK1A
SCHEMBL4005872 0.71 PDPK1 (0.40) BRAFTNNI3KMAPK1CHEK1IRAK4
SCHEMBL6469764 0.70 BRAF (0.43) BRAFTNNI3KMAPK1CHEK1IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed