SCHEMBL4007170

SCHEMBL4007170

Brc1c[nH]c2ncnc(-c3ccccc3)c12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 9/20 0.55
JAK3 P52333 9/20 0.55
ROCK2 O75116 5/20 0.48
LIMK1 P53667 5/20 0.48
LRRK2 Q5S007 5/20 0.47
PRKACA P17612 5/20 0.44
GSK3A P49840 5/20 0.44
GSK3B P49841 5/20 0.44
CDK5 Q00535 5/20 0.44
ROCK1 Q13464 5/20 0.44
DYRK1A Q13627 5/20 0.44
PRKD3 O94806 4/20 0.44
MAP4K4 O95819 4/20 0.44
CLK2 P49760 4/20 0.44
MAP4K2 Q12851 4/20 0.44
NTRK1 P04629 4/20 0.44
TAOK1 Q7L7X3 3/20 0.44
CLK4 Q9HAZ1 3/20 0.44
NTRK3 Q16288 3/20 0.44
NTRK2 Q16620 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15032780 0.83 KIT (0.44) JAK2JAK3DYRK1ANTRK1KIT
SCHEMBL15032863 0.81 JAK3 (0.68) JAK2JAK3ROCK2LIMK1LRRK2
SCHEMBL20195296 0.80 LIMK1 (0.69) JAK2JAK3ROCK2LIMK1LRRK2
SCHEMBL15010414 0.80 JAK2 (0.55) JAK2JAK3ROCK2LIMK1LRRK2
SCHEMBL15032846 0.77 PIK3CD (0.46) JAK2JAK3
SCHEMBL20184432 0.76 JAK3 (0.68) JAK2JAK3ROCK2LIMK1
SCHEMBL4006360 0.75 BRAF (0.60) ROCK2LIMK1LRRK2PRKACAGSK3B
SCHEMBL20184454 0.74 JAK3 (0.70) JAK2JAK3ROCK2LIMK1
SCHEMBL4790325 0.73 LRRK2 (0.61) JAK2JAK3ROCK2LIMK1LRRK2
SCHEMBL15032654 0.71 JAK3 (1.00) JAK2JAK3ROCK2LIMK1LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed