SCHEMBL4007696

SCHEMBL4007696

CCCCOC(=O)N1CCC(COC(C)c2cc(Cl)cc3c(Br)n[nH]c23)(c2ccc(F)cc2)CC1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CTSK P43235 1/20 0.35
OPRD1 P41143 2/20 0.34
OPRK1 P41145 1/20 0.34
SMYD3 Q9H7B4 1/20 0.33
HRH2 P25021 1/20 0.31
HRH1 P35367 1/20 0.31
MCHR1 Q99705 1/20 0.31
ENPP2 Q13822 3/20 0.31
ATXN2 Q99700 3/20 0.31
S1PR2 O95136 1/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4014639 0.93 CTSK (0.35) CTSKOPRD1OPRK1HRH2HRH1
SCHEMBL12290809 0.87 TACR1 (0.38) CYP3A4
SCHEMBL2424821 0.87 TACR1 (0.38) CYP3A4
SCHEMBL2428449 0.87 TACR1 (0.38) CYP3A4
SCHEMBL2425742 0.84 TACR1 (0.41)
SCHEMBL2425740 0.84 TACR1 (0.41)
SCHEMBL2425829 0.81 TACR1 (0.39)
SCHEMBL2425826 0.81 TACR1 (0.39)
SCHEMBL2427521 0.81 TACR1 (0.33) CTSKS1PR2
SCHEMBL2427706 0.81 TACR1 (0.33) CTSKENPP2ATXN2S1PR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009009411-A1 SUBSTITUTED HETEROCYCLIC ETHERS AND THEIR USE IN CNS DISORDERS BRISTOL-MYERS SQUIBB COMPANY (US) 2009-01-15 WO disclosed