SCHEMBL4007925

SCHEMBL4007925

CCCc1nc(=O)c(Oc2cccc3c2OC(C)(C)C3)c(CC)n1Cc1ccc(-c2ccccc2C#N)cc1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.47
ACHE P22303 1/20 0.38
AGTR1 P30556 2/20 0.36
APLNR P35414 1/20 0.35
AGTR2 P50052 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1886189 0.89 PPARG (0.47) PPARGACHEAGTR1APLNRAGTR2
SCHEMBL4016260 0.81 PPARG (0.52) PPARGACHEAGTR1
SCHEMBL4012577 0.80 PPARG (0.57) PPARGACHEAGTR1AGTR2
SCHEMBL4010050 0.80 PPARG (0.49) PPARGACHEAGTR1AGTR2
SCHEMBL4016898 0.79 PPARG (0.54) PPARGACHEAGTR1
SCHEMBL4007590 0.78 PPARG (0.53) PPARGACHEAGTR1
SCHEMBL4012893 0.78 PPARG (0.51) PPARGACHEAGTR1AGTR2
SCHEMBL4009893 0.77 PPARG (0.51) PPARGAGTR1APLNRAGTR2
SCHEMBL4013600 0.77 PPARG (0.49) PPARGACHEAGTR1AGTR2
SCHEMBL4010668 0.76 PPARG (0.63) PPARGACHEAGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009133970-A1 CRYSTALLINE COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-05 WO disclosed
EP-2074117-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2009-07-01 EP disclosed
WO-2008062905-A2 HETEROMONOCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-05-29 WO disclosed