SCHEMBL4009713

SCHEMBL4009713

CSc1c(C)[nH]c2nc(C)ccc12

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.45
KMT2A Q03164 2/20 0.45
ADORA1 P30542 7/20 0.41
ADORA2A P29274 6/20 0.41
PDK2 Q15119 1/20 0.40
PDK4 Q16654 1/20 0.40
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13959224 0.81 ADORA2A (0.43) KMT2AADORA1ADORA2A
SCHEMBL29814700 0.74 KDM4E (0.46) KDM4EKMT2AADORA1ADORA2APDK2
SCHEMBL23089134 0.74 KDM4E (0.46) KDM4EKMT2AADORA1ADORA2APDK2
SCHEMBL23132920 0.72 ADORA1 (0.46) KDM4EKMT2AADORA1ADORA2APDK2
SCHEMBL24859522 0.72 KDM4E (0.44) KDM4EKMT2AADORA1ADORA2APDK2
SCHEMBL23103525 0.72 KDM4E (0.44) KDM4EKMT2AADORA1ADORA2APDK2
SCHEMBL19249730 0.69 CCR1 (0.41) KMT2AMEN1
SCHEMBL23106887 0.69 ADORA1 (0.55) KDM4EKMT2AADORA1ADORA2APDK2
SCHEMBL8324036 0.68 IDO1 (0.38) KDM4EKMT2AADORA1ADORA2AMEN1
SCHEMBL9695650 0.67 HTT (0.51) KDM4EKMT2AADORA1ADORA2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009005672-A1 ANTIDIABETIC AZAINDOLES AND DIAZAINDOLES MERCK & CO., INC. (US) 2009-01-08 WO disclosed
WO-2009005672-A1 ANTIDIABETIC AZAINDOLES AND DIAZAINDOLES MERCK & CO., INC. (US) 2009-01-08 WO disclosed