SCHEMBL401001

SCHEMBL401001

[CH2]c1cccc(N(CC)CC)c1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.59
CYP3A4 P08684 2/20 0.59
TERT O14746 1/20 0.44
S100B P04271 1/20 0.42
TSHR P16473 2/20 0.41
L3MBTL1 Q9Y468 5/20 0.40
MAPK1 P28482 3/20 0.40
RECQL P46063 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
PSMD14 O00487 1/20 0.40
GFER P55789 1/20 0.40
KMT2A Q03164 4/20 0.39
MAPT P10636 3/20 0.39
MEN1 O00255 3/20 0.39
GAA P10253 3/20 0.39
NPC1 O15118 1/20 0.39
GRK6 P43250 1/20 0.39
RAB9A P51151 1/20 0.39
HIF1A Q16665 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1574035 0.84 ALDH1A1 (0.71) ALDH1A1CYP3A4TERTS100BTSHR
SCHEMBL7335494 0.83 ALDH1A1 (0.41) ALDH1A1CYP3A4MAPTALDH3A1ALDH1A3
SCHEMBL2091963 0.81 ALDH1A1 (0.38) ALDH1A1CYP3A4TSHRGLA
SCHEMBL297874 0.77 ALDH1A1 (0.41) ALDH1A1CYP3A4TERTS100BTSHR
SCHEMBL30565135 0.76 ALDH1A1 (0.61) ALDH1A1CYP3A4TERTS100BTSHR
SCHEMBL457496 0.76 ALDH1A1 (0.61) ALDH1A1CYP3A4TERTS100BTSHR
SCHEMBL30565134 0.76 ALDH1A1 (0.61) ALDH1A1CYP3A4TERTS100BTSHR
SCHEMBL14283564 0.76 ALDH1A1 (0.61) ALDH1A1CYP3A4TERTS100BTSHR
SCHEMBL3425607 0.76 ALDH1A1 (0.61) ALDH1A1CYP3A4TERTS100BTSHR
SCHEMBL11638767 0.76 ALDH1A1 (0.61) ALDH1A1CYP3A4TERTS100BTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 43 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815108-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-01-07 EP claimed
US-5683999-A Cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-04 US claimed
WO-1996029329-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-26 WO claimed
CN-108117551-B Substituted (1H-pyrazolo [3,4-b ] pyridine) urea compound and anti-tumor application thereof 华东理工大学 2020-03-27 CN disclosed
US-8729262-B2 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2014-05-20 US disclosed
US-8318738-B2 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2012-11-27 US disclosed
US-8138337-B2 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2012-03-20 US disclosed
CN-1942472-B Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORP. (KR) 2012-02-15 CN disclosed
US-8106049-B2 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2012-01-31 US disclosed
US-8101751-B2 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2012-01-24 US disclosed
US-8049008-B2 Reverse-turn mimetics and method relating thereto CHOONGWAE PHARMA CORPORATION (KR) 2011-11-01 US disclosed
US-5683999-A Cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-04 US disclosed
US-5591714-A TREATING VANCOMYCIN RESISTANT ENTEROCOCCUS INFECTIONS WITH GLYCOPEPTIDE ANTIBIOTIC ELI LILLY AND COMPANY (US) 1997-01-07 US disclosed
WO-1996029329-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-09-26 WO disclosed
EP-0239129-B1 HYDROQUINOLINE COMPOUNDS, COMPOSITIONS CONTAINING SAME AND PROCESSES FOR PREPARING SAME OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1991-09-25 EP disclosed
EP-0435503-A1 Improvements in or relating to gylcopeptide derivatives ELI LILLY AND COMPANY (US) 1991-07-03 EP disclosed
US-4963566-A ANTIULCER AGENT OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-10-16 US disclosed
EP-0239129-A2 Hydroquinoline compounds, compositions containing same and processes for preparing same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1987-09-30 EP disclosed
US-3980660-A ANTIAUERGENS, ANAPHYLACTIC THE UPJOHN COMPANY (US) 1976-09-14 US disclosed
US-3972911-A PROPHYLAXIS THE UPJOHN COMPANY (US) 1976-08-03 US disclosed