SCHEMBL4010315

SCHEMBL4010315

Cc1cnc2c(Br)cccc2c1-c1cccc(O)c1

nearest known ligand 0.46

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 18/20 0.46
NR1H3 Q13133 16/20 0.46
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
HSD17B1 P14061 1/20 0.41
HSD17B2 P37059 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL35460 0.83 NR1H2 (0.61) NR1H2NR1H3HSD17B1HSD17B2
SCHEMBL35135 0.81 NR1H2 (0.64) NR1H2NR1H3
SCHEMBL4012944 0.74 NR1H2 (0.79) NR1H2NR1H3
SCHEMBL1125162 0.72 NR1H2 (0.58) NR1H2NR1H3
SCHEMBL1125801 0.72 NR1H2 (0.52) NR1H2NR1H3
SCHEMBL4011832 0.70 NR1H2 (0.64) NR1H2NR1H3
SCHEMBL1125912 0.69 NR1H2 (0.52) NR1H2NR1H3
SCHEMBL2766777 0.69 ALDH1A1 (0.48) NR1H2NR1H3MAPT
SCHEMBL1125269 0.68 NR1H2 (0.53) NR1H2NR1H3
SCHEMBL1125990 0.68 NR1H2 (0.50) NR1H2NR1H3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2074098-A2 QUINOLINE COMPOUNDS Wyeth (US) 2009-07-01 EP disclosed
WO-2008049047-A2 QUINOLINE COMPOUNDS WYETH (US) 2008-04-24 WO disclosed