SCHEMBL4010493

SCHEMBL4010493

O=C(Cn1cc(-c2ccccc2Cl)c2c(-c3ccccc3)ncnc21)N1CCC(n2c(=O)[nH]c3ncccc32)CC1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CALCRL Q16602 19/20 0.56
TNKS O95271 1/20 0.46
PARP1 P09874 1/20 0.46
PARP2 Q9UGN5 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4010288 0.95 CALCRL (0.54) CALCRL
SCHEMBL4003427 0.90 CALCRL (0.57) CALCRLTNKSPARP1PARP2
SCHEMBL4006748 0.89 CALCRL (0.56) CALCRLTNKSPARP1PARP2
SCHEMBL4008402 0.89 CALCRL (0.56) CALCRLTNKSPARP1PARP2
SCHEMBL13769399 0.88 CALCRL (0.54) CALCRL
SCHEMBL4005494 0.88 CALCRL (0.55) CALCRL
SCHEMBL4013384 0.88 CALCRL (0.57) CALCRLTNKSPARP1PARP2
SCHEMBL13769952 0.88 CALCRL (0.57) CALCRLTNKSPARP1PARP2
SCHEMBL4007640 0.88 CALCRL (0.55) CALCRLTNKSPARP1PARP2
SCHEMBL13769702 0.87 CALCRL (0.55) CALCRLTNKSPARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed
WO-2009080682-A1 PYRROLO[2,3-D]PYRIMIDINE DERIVATIVES AS CGRP RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2009-07-02 WO disclosed