SCHEMBL4010938

SCHEMBL4010938

O=C(O)N1CCc2ccc(CI)cc2C1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43
NPC1 O15118 5/20 0.42
RAB9A P51151 3/20 0.42
KMT2A Q03164 5/20 0.41
TMEM97 Q5BJF2 2/20 0.41
SIGMAR1 Q99720 2/20 0.41
NOTUM Q6P988 1/20 0.41
ALDH1A1 P00352 2/20 0.40
PDE4B Q07343 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
NR1H2 P55055 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
MEN1 O00255 3/20 0.40
MAPT P10636 1/20 0.40
TAAR1 Q96RJ0 1/20 0.40
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27914873 0.86 NAMPT (0.49) ESR1ESR2NPC1RAB9AKMT2A
SCHEMBL22981196 0.85 ESR1 (0.43) ESR1ESR2NPC1RAB9AKMT2A
SCHEMBL27933360 0.82 NPC1 (0.43) ESR1ESR2NPC1RAB9AKMT2A
SCHEMBL4019716 0.81 ESR1 (0.41) ESR1ESR2NPC1RAB9AKMT2A
SCHEMBL16634622 0.80 NAMPT (0.49) ESR1ESR2NPC1RAB9AKMT2A
SCHEMBL4015963 0.80 NR1H2 (0.67) ESR1ESR2NPC1RAB9ATMEM97
SCHEMBL19717635 0.79 NPC1 (0.45) ESR1ESR2NPC1RAB9AKMT2A
SCHEMBL1648634 0.78 ESR2 (0.68) ESR1ESR2KMT2ANOTUMNR1H2
SCHEMBL30199245 0.78 ESR2 (0.68) ESR1ESR2KMT2ANOTUMNR1H2
SCHEMBL28675076 0.77 TMEM97 (0.43) ESR1ESR2NPC1KMT2ATMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2044017-A2 SUBSTITUTED PHENYL ACETIC ACIDS AS DP-2 ANTAGONISTS ICOS CORPORATION (US) 2009-04-08 EP disclosed
WO-2007146838-A2 SUBSTITUTED PHENYL ACETIC ACIDS AS DP-2 ANTAGONISTS ICOS CORPORATION (US) 2007-12-21 WO disclosed